SCHEMBL790485

SCHEMBL790485

O=C(c1nc(Nc2ccccc2F)sc1F)N1CCc2ccccc2C1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.55
RAB9A P51151 5/20 0.55
TRPC3 Q13507 2/20 0.51
TRPC6 Q9Y210 2/20 0.51
HPGD P15428 3/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
MEN1 O00255 1/20 0.47
LMNA P02545 1/20 0.47
ALOX12 P18054 1/20 0.47
NFKB1 P19838 1/20 0.47
NFKB2 Q00653 1/20 0.47
KMT2A Q03164 1/20 0.47
RELA Q04206 1/20 0.47
ALDH1A1 P00352 3/20 0.45
PDE4B Q07343 2/20 0.44
PDE4D Q08499 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
CTDSP1 Q9GZU7 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
MAOB P27338 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10080532 0.90 TRPC3 (0.54) NPC1RAB9ATRPC3TRPC6HPGD
SCHEMBL10080530 0.90 TRPC3 (0.63) NPC1RAB9ATRPC3TRPC6HPGD
SCHEMBL806828 0.81 TRPC3 (0.64) NPC1RAB9ATRPC3TRPC6HPGD
SCHEMBL10080527 0.80 TRPC3 (0.66) NPC1RAB9ATRPC3TRPC6HPGD
SCHEMBL10080531 0.77 TRPC3 (0.58) NPC1RAB9ATRPC3TRPC6HPGD
SCHEMBL807012 0.77 TRPC3 (0.62) NPC1RAB9ATRPC3TRPC6HPGD
SCHEMBL10080528 0.73 RAB9A (0.58) NPC1RAB9ATRPC3TRPC6HPGD
SCHEMBL10080529 0.70 TRPC3 (0.58) NPC1RAB9ATRPC3TRPC6HPGD
SCHEMBL4923910 0.69 KDM4E (0.58) NPC1RAB9ATRPC3TRPC6HPGD
SCHEMBL798510 0.68 TRPC3 (0.67) NPC1RAB9ATRPC3TRPC6HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037349-A2 COMPOUNDS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed
WO-2012037349-A2 COMPOUNDS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed