SCHEMBL7904903

SCHEMBL7904903

COc1cccc(CC(C)(C)OC(=O)C(O)C2CCNCC2)c1OC

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 2/20 0.38
TP53 P04637 1/20 0.38
KMT2A Q03164 2/20 0.36
GNAI3 P08754 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6989780 0.76 SLC6A2 (0.46) SLC6A2SLC6A4ALDH1A1KDM4ETP53
Trifluoroacetamide SCHEMBL6993217 0.74 SLC6A2 (0.40) SLC6A2SLC6A4ALDH1A1KDM4ETP53
Methanesulfonamide SCHEMBL6999861 0.72 CA2 (0.44) SLC6A2SLC6A4ALDH1A1TP53GNAI3
SCHEMBL8105808 0.69 MMP13 (0.39) SLC6A2SLC6A4KMT2A
SCHEMBL3048145 0.68 HTR2C (0.55) SLC6A2SLC6A4
SCHEMBL13701283 0.68 HTR2C (0.55) SLC6A2SLC6A4
SCHEMBL3048141 0.68 HTR2C (0.55) SLC6A2SLC6A4
SCHEMBL4225398 0.68 HTR2C (0.55) SLC6A2SLC6A4
SCHEMBL412203 0.68 CPN1 (0.36) SLC6A2SLC6A4TSHR
Trifluoroacetamide SCHEMBL6991362 0.68 L3MBTL1 (0.36) SLC6A2SLC6A4ALDH1A1KDM4ETP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1107753-A1 MULTIVALENT AGONISTS, PARTIAL AGONISTS, INVERSE AGONISTS AND ANTAGONISTS OF THE 5HT2 RECEPTORS Advanced Medicine, Inc. (US) 2001-06-20 EP disclosed
EP-1082289-A4 METHODS FOR IDENTIFYING NOVEL MULTIMERIC AGENTS THAT MODULATE RECEPTORS ADVANCED MEDICINE INC (US) 2001-03-14 EP disclosed
EP-1082289-A1 METHODS FOR IDENTIFYING NOVEL MULTIMERIC AGENTS THAT MODULATE RECEPTORS Advanced Medicine, Inc. (US) 2001-03-14 EP disclosed
WO-1999066944-A9 METHODS FOR IDENTIFYING NOVEL MULTIMERIC AGENTS THAT MODULATE RECEPTORS ADVANCED MEDICINE INC (US) 2000-07-27 WO disclosed
WO-1999066944-A1 METHODS FOR IDENTIFYING NOVEL MULTIMERIC AGENTS THAT MODULATE RECEPTORS ADVANCED MEDICINE, INC. (US) 1999-12-29 WO disclosed
WO-1999063996-A1 MULTIVALENT AGONISTS, PARTIAL AGONISTS, INVERSE AGONISTS AND ANTAGONISTS OF THE 5HT2 RECEPTORS ADVANCED MEDICINE, INC. (US) 1999-12-16 WO disclosed