SCHEMBL7905274

SCHEMBL7905274

CN(C)CCOc1ccccc1-c1nnc(-n2nc(N3CCCCC3)nc2N)s1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 5/20 0.41
HTR7 P34969 2/20 0.38
NOS3 P29474 5/20 0.38
NOS1 P29475 5/20 0.38
NOS2 P35228 5/20 0.38
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PIK3CD O00329 1/20 0.33
PIK3R1 P27986 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CB P42338 1/20 0.33
ADRB2 P07550 1/20 0.33
ADRB1 P08588 1/20 0.33
HTR1B P28222 1/20 0.33
SYK P43405 1/20 0.33
PTPN11 Q06124 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7902674 0.96 HRH3 (0.40) HRH3HTR7NOS3NOS1NOS2
SCHEMBL7904622 0.95 HRH3 (0.39) HRH3HTR7NOS3NOS1NOS2
SCHEMBL7896508 0.88 HRH3 (0.41) HRH3KDM4EALDH1A1PTPN11
SCHEMBL7905780 0.87 HRH3 (0.40) HRH3KDM4EALDH1A1PTPN11
SCHEMBL7902706 0.87 HRH3 (0.38) HRH3KDM4EALDH1A1HTR1B
SCHEMBL7904665 0.87 HRH3 (0.36) HRH3KDM4EALDH1A1SMN1; SMN2
SCHEMBL7908481 0.87 PIK3CB (0.44) HRH3KDM4EPIK3CDPIK3R1PIK3CA
SCHEMBL7896504 0.86 HRH3 (0.39) HRH3HTR7KDM4EALDH1A1PTPN11
SCHEMBL7896424 0.83 ALDH1A1 (0.42) HRH3KDM4EALDH1A1SMN1; SMN2
SCHEMBL7896433 0.82 POLB (0.38) KDM4EALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6191152-B1 CARDIOVASCULAR DISORDERS, NERVOUS SYSTEM DISORDERS EGIS GYÓGYSZERGYAR RT. (HU) 2001-02-20 US disclosed