SCHEMBL790597

SCHEMBL790597

COc1cc(Br)ccc1-c1c(N)nc2ccc(I)cc2c1C#N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 4/20 0.39
ADORA2A P29274 3/20 0.39
EGFR P00533 2/20 0.38
ERBB2 P04626 1/20 0.38
KDM4E B2RXH2 4/20 0.38
ALDH1A1 P00352 4/20 0.38
HPGD P15428 1/20 0.38
DHFR P00374 2/20 0.36
STK10 O94804 1/20 0.36
SLK Q9H2G2 1/20 0.36
HSD17B10 Q99714 1/20 0.35
APP P05067 1/20 0.35
GSK3A P49840 1/20 0.35
GSK3B P49841 1/20 0.35
DYRK1A Q13627 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
ABCC8 Q09428 1/20 0.34
KCNJ11 Q14654 1/20 0.34
MEN1 O00255 1/20 0.34
GLA P06280 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL790927 0.84 APP (0.37) EGFRAPPGAAMAPT
SCHEMBL10277683 0.80 SIK1 (0.39) KDM4EALDH1A1HPGDAPPMEN1
SCHEMBL790759 0.73 KDM4E (0.47) ADORA1ADORA2AKDM4EALDH1A1HPGD
SCHEMBL1414662 0.66 ADORA1 (0.39) ADORA1ADORA2AKDM4EALDH1A1HPGD
SCHEMBL790933 0.66 APP (0.47) ADORA2AKDM4EALDH1A1HPGDDHFR
SCHEMBL790839 0.65 ADORA2A (0.49) ADORA1ADORA2AKDM4EALDH1A1HPGD
SCHEMBL7913439 0.65 KDM4E (0.60) ADORA1ADORA2AEGFRKDM4EALDH1A1
SCHEMBL6223729 0.64 ALDH1A1 (0.67) ADORA1ADORA2AKDM4EALDH1A1HPGD
SCHEMBL27576309 0.64 ADORA1 (0.55) ADORA1ADORA2AEGFRERBB2KDM4E
SCHEMBL27470171 0.61 ADORA2A (0.58) ADORA1ADORA2AKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed