SCHEMBL790839

SCHEMBL790839

N#Cc1c(-c2ccc(N3CCOCC3)cc2)c(N)nc2ccc(I)cc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.49
CCNA2 P20248 3/20 0.44
CDK2 P24941 3/20 0.44
CDK1 P06493 1/20 0.41
CDK4 P11802 1/20 0.41
CCNB1 P14635 1/20 0.41
CCND1 P24385 1/20 0.41
CDK7 P50613 1/20 0.41
CCNH P51946 1/20 0.41
MAPT P10636 5/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
TP53 P04637 1/20 0.40
ALOX15 P16050 1/20 0.40
KDM4E B2RXH2 6/20 0.40
ALDH1A1 P00352 3/20 0.40
HTT P42858 3/20 0.40
LMNA P02545 3/20 0.40
HPGD P15428 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL789847 0.85 JAK2 (0.46) ADORA2ACDK1SMN1; SMN2KDM4EALDH1A1
SCHEMBL790716 0.83 MAPT (0.43) ADORA2AMAPTSMN1; SMN2NPC1RAB9A
SCHEMBL790759 0.81 KDM4E (0.47) ADORA2ASMN1; SMN2KDM4EALDH1A1HTT
SCHEMBL10277681 0.80 LRRK2 (0.47) MAPTSMN1; SMN2NPC1RAB9ATP53
SCHEMBL10277093 0.78 KDM4E (0.43) ADORA2ACCNA2CDK2CDK1CDK4
SCHEMBL940196 0.75 ADORA2A (0.50) ADORA2AMAPTSMN1; SMN2NPC1RAB9A
SCHEMBL940655 0.75 ADORA2A (0.47) ADORA2ACDK2CDK1MAPTSMN1; SMN2
SCHEMBL9954672 0.69 TDO2 (0.52) MAPTSMN1; SMN2NPC1RAB9ATP53
SCHEMBL790084 0.69 JAK2 (0.48) SMN1; SMN2KDM4EALDH1A1HPGD
SCHEMBL941557 0.68 PIK3CB (0.50) ADORA2AMAPTSMN1; SMN2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed