SCHEMBL7909124

SCHEMBL7909124

Cc1noc(-c2ccc(C(=O)N3CCC(C(=O)N[C@@H](C)C4=CC=CCC4)(C4=CC=CCC4)CC3)cc2)n1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 2/20 0.34
TACR3 P29371 3/20 0.33
GPR119 Q8TDV5 1/20 0.33
CYP3A4 P08684 3/20 0.32
KCNH2 Q12809 2/20 0.32
CYP1A2 P05177 2/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
TBK1 Q9UHD2 4/20 0.32
ALDH1A1 P00352 2/20 0.32
FASN P49327 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
IKBKE Q14164 1/20 0.31
LMNA P02545 1/20 0.30
MGLL Q99685 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7910233 0.80 CYP3A4 (0.34) CYP3A4CYP1A2CYP2C19ALDH1A1
SCHEMBL7908120 0.79 MGLL (0.42) ALDH1A1HDAC4HDAC2HDAC8HDAC6
SCHEMBL7908118 0.78 ALDH1A1 (0.45) GPR119CYP3A4ALDH1A1
SCHEMBL7906027 0.77 ACACB (0.32) CYP3A4
SCHEMBL7915500 0.76 ALDH1A1 (0.42) ALDH1A1FASNMGLL
SCHEMBL378915 0.76 TSHR (0.43) BDKRB1TBK1ALDH1A1MGLL
SCHEMBL7910802 0.76 TSHR (0.39) ALDH1A1FASN
SCHEMBL7913727 0.76 KDM4E (0.37) CYP3A4ALDH1A1LMNA
SCHEMBL379355 0.75 TACR3 (0.41) BDKRB1TACR3CYP1A2CYP2C9CYP2C19
SCHEMBL7902201 0.74 RAB9A (0.48) TACR3CYP3A4KCNH2CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010106081-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-23 WO disclosed