SCHEMBL7909779

SCHEMBL7909779

O=c1[nH]cc(C(F)(F)F)cc1Br

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
GLA P06280 1/20 0.44
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
HPGD P15428 2/20 0.39
LMNA P02545 1/20 0.38
DAO P14920 5/20 0.37
ERCC1 P07992 1/20 0.36
ERCC4 Q92889 1/20 0.36
ACLY P53396 1/20 0.35
PARP1 P09874 1/20 0.35
HSD17B10 Q99714 1/20 0.33
CYP1A2 P05177 1/20 0.32
ALOX12 P18054 1/20 0.32
CBLB Q13191 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14155894 0.79 ALDH1A1 (0.44) ALDH1A1GLAHPGDDAOERCC1
SCHEMBL17002554 0.77 MEN1 (0.48) ALDH1A1MEN1KMT2AHPGDLMNA
SCHEMBL17362093 0.77 ACLY (0.42) ALDH1A1MEN1KMT2AHPGDLMNA
SCHEMBL574325 0.75 TTK (0.44) ALDH1A1GLAMEN1KMT2AHPGD
SCHEMBL4153740 0.75 PKM (0.54) ALDH1A1MEN1KMT2AHPGDLMNA
SCHEMBL1000301 0.75 DAO (0.50) ALDH1A1MEN1KMT2AHPGDLMNA
SCHEMBL6986501 0.75 DAO (0.40) ALDH1A1MEN1KMT2AHPGDLMNA
SCHEMBL29291942 0.73 MEN1 (0.31) ALDH1A1MEN1KMT2AHPGD
SCHEMBL25651305 0.72 ALDH1A1 (0.47) ALDH1A1MEN1KMT2AHPGDLMNA
SCHEMBL9730796 0.72 MEN1 (0.38) ALDH1A1MEN1KMT2AHPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4546191-A Trifluoromethyl-2-pyridinone or pyridinthione compounds and process for the preparation of the same ISHIHARA SANGYO KAISHA LTD. (JP) 1985-10-08 US claimed
US-20250163038-A1 CBL-B MODULATORS AND USES THEREOF NIMBUS CLIO, INC. 2025-05-22 US disclosed
EP-4359381-A1 CBL-B MODULATORS AND USES THEREOF Nimbus Clio, Inc. (US) 2024-05-01 EP disclosed
CN-117858865-A CBL-B modulators and uses thereof 林伯士克莱奥公司 2024-04-09 CN disclosed
WO-2022272248-A1 CBL-B MODULATORS AND USES THEREOF NIMBUS CLIO, INC. (US) 2022-12-29 WO disclosed
WO-2022272248-A1 CBL-B MODULATORS AND USES THEREOF NIMBUS CLIO, INC. (US) 2022-12-29 WO disclosed
CN-107074828-B Compounds and compositions as RAF kinase inhibitors 诺华股份有限公司 2020-05-19 CN disclosed
EP-3239147-B1 QUINOLINE DERIVATIVE ONO PHARMACEUTICAL CO (JP) 2019-08-28 EP disclosed
EP-3191478-B1 COMPOUNDS AND COMPOSITIONS AS RAF KINASE INHIBITORS NOVARTIS AG (CH) 2019-05-08 EP disclosed
US-10208034-B2 Quinoline derivative ONO PHARMACEUTICAL CO., LTD. (JP) 2019-02-19 US disclosed
WO-1998054187-A1 SPIRO-AZACYCLIC DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LIMITED (GB) 1998-12-03 WO disclosed
EP-0880501-A1 HETEROCYCLIC COMPOUNDS USEFUL AS PHARMACEUTICAL AGENTS ZENECA LIMITED (GB) 1998-12-02 EP disclosed
WO-1997028128-A1 HETEROCYCLIC COMPOUNDS USEFUL AS PHARMACEUTICAL AGENTS ZENECA LIMITED (GB) 1997-08-07 WO disclosed
US-5109004-A Cyano phenyl-substituted with heterocylic compound; insecticides, miticides IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-04-28 US disclosed
EP-0398499-A2 Insecticides ZENECA LIMITED (GB) 1990-11-22 EP disclosed
CN-1046526-A New compound and preparation method thereof ICI PLC (GB) 1990-10-31 CN disclosed
EP-0367410-A1 Aryl pyridones as insecticidal agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-05-09 EP disclosed
EP-0272824-A2 Chemical compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-06-29 EP disclosed
CN-86106734-A ARYL PYRIDONES 1987-04-01 CN disclosed
US-4546191-A Trifluoromethyl-2-pyridinone or pyridinthione compounds and process for the preparation of the same ISHIHARA SANGYO KAISHA LTD. (JP) 1985-10-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250163038-A1 CBL-B MODULATORS AND USES THEREOF CBLB, CBL, CBLC ALDH1A1 4185/4885GLA 2765/4885MEN1 4401/4885
US-10208034-B2 Quinoline derivative FLT3, AXL, ABL1 ALDH1A1 3586/4885GLA 1239/4885MEN1 441/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.