SCHEMBL7909970

SCHEMBL7909970

FC(F)(F)COc1ncc(-n2ccnc2C(F)(F)F)cc1Br

nearest known ligand 0.35

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.35
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7919399 0.85 S100A9 (0.35)
SCHEMBL7916846 0.78 CHRNB2 (0.42)
SCHEMBL7919587 0.72 CHRNB2 (0.46)
SCHEMBL8149329 0.72 PTGS2 (0.42) PTGS2
SCHEMBL7917315 0.70 PTGS2 (0.48) ADORA2APTGS2
SCHEMBL8118971 0.70 MAPT (0.36) PTGS2
SCHEMBL8177172 0.69 NR1I2 (0.35) PTGS2
SCHEMBL14823453 0.69 PTGS2 (0.38) ADORA2APTGS2
SCHEMBL2114332 0.69 MAPT (0.46) ADORA2APTGS2
SCHEMBL29837825 0.69 L3MBTL1 (0.38) ADORA2APTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6225320-B1 TREATMENT OF PAIN, INFLAMMATION, MIGRAINE, EMESIS AND POSTTHERPETIC NEURALGIA MERCK SHARP & DOHME LTD. (GB) 2001-05-01 US disclosed