SCHEMBL7919587

SCHEMBL7919587

COc1cc(-n2ccnc2C(F)(F)F)cnc1Br

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 9/20 0.46
CHRNA4 P43681 9/20 0.46
CHRNB4 P30926 7/20 0.41
CHRNA3 P32297 7/20 0.41
NR1I2 O75469 1/20 0.33
HSD11B1 P28845 1/20 0.33
TSHR P16473 1/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
KMT2A Q03164 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
PTK2 Q05397 1/20 0.31
TUBB4A P04350 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7919399 0.81 S100A9 (0.35) NR1I2HSD11B1KDM4EMEN1ALDH1A1
SCHEMBL8149329 0.78 PTGS2 (0.42) NR1I2HSD11B1HTTSMN1; SMN2KDM4E
SCHEMBL7916641 0.75 CHRNB2 (0.45) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL7916846 0.73 CHRNB2 (0.42) CHRNB2CHRNA4NR1I2HSD11B1HTT
SCHEMBL7919134 0.73 ALDH1A1 (0.33) TSHRHTTSMN1; SMN2KDM4EMEN1
SCHEMBL7909970 0.72 ADORA2A (0.35)
SCHEMBL9080396 0.71 ALDH1A1 (0.45) TSHRHTTSMN1; SMN2KDM4EMEN1
SCHEMBL31045735 0.70 CHRNB2 (0.43) CHRNB2CHRNA4CHRNB4CHRNA3TSHR
SCHEMBL8118971 0.68 MAPT (0.36) NR1I2HSD11B1HTTSMN1; SMN2KDM4E
SCHEMBL8177172 0.68 NR1I2 (0.35) NR1I2HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6225320-B1 TREATMENT OF PAIN, INFLAMMATION, MIGRAINE, EMESIS AND POSTTHERPETIC NEURALGIA MERCK SHARP & DOHME LTD. (GB) 2001-05-01 US disclosed