SCHEMBL7911295

SCHEMBL7911295

CC1=CN2C=C(Cc3ccc(NC(N)=O)cc3)C=C(c3cccc(Cl)c3)C2N1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 1/20 0.48
KMT2A Q03164 2/20 0.35
RORC P51449 2/20 0.35
MEN1 O00255 1/20 0.35
PRKD3 O94806 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
PRKD1 Q15139 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PRKD2 Q9BZL6 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PDE4B Q07343 5/20 0.34
FGFR3 P22607 1/20 0.34
KDR P35968 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
PLAU P00749 1/20 0.33
IKBKB O14920 1/20 0.33
NPC1 O15118 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7916616 0.85 PDE4D (0.48) PDE4DKMT2ARORCMEN1PRKD3
SCHEMBL7913253 0.85 MAOB (0.34) ALDH1A1SMN1; SMN2PDE4BCYP3A4CYP2C19
SCHEMBL7914652 0.82 DYRK3 (0.37) KMT2AMEN1ALDH1A1
SCHEMBL7902852 0.80 NPC1 (0.34) KMT2ASMN1; SMN2NPC1
SCHEMBL7912990 0.79 PARP1 (0.37) KMT2AMEN1ALDH1A1
SCHEMBL7913078 0.79 DYRK3 (0.37)
SCHEMBL7917981 0.79 DYRK3 (0.35) KMT2AMEN1ALDH1A1
SCHEMBL7929296 0.79 DYRK3 (0.49) ALDH1A1SMN1; SMN2
SCHEMBL7911686 0.78 PGR (0.34) KMT2AMEN1ALDH1A1HPGDSMN1; SMN2
SCHEMBL7902988 0.77 GRIN1 (0.32) PDE4DSMN1; SMN2CYP3A4CYP2C19NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059838-A2 PDE4 INHIBITORS SELECTIVE FOR THE LONG FORM OF PDE4 FOR TREATING INFLAMMATION AND AVOIDING SIDE EFFECTS DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed
WO-2010059836-A1 SUBSTITUTED AZA-BRIDGED BICYCLICS FOR CARDIOVASCULAR AND CNS DISEASE DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed