SCHEMBL7912645

SCHEMBL7912645

Bc1ccnc(N)c1C#N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKACA P17612 2/20 0.38
PRKACG P22612 2/20 0.38
PRKACB P22694 2/20 0.38
LRRK2 Q5S007 2/20 0.36
NOS3 P29474 3/20 0.34
NOS2 P35228 3/20 0.34
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GLA P06280 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
KMT2A Q03164 1/20 0.33
ABL1 P00519 1/20 0.33
ADORA2A P29274 6/20 0.33
ADORA1 P30542 6/20 0.33
ADORA2B P29275 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19139283 0.79 NOS3 (0.34) NOS3NOS2F12PLAUNCF1
SCHEMBL27427296 0.78 PRKACA (0.46) PRKACAPRKACGPRKACBLRRK2NOS3
SCHEMBL15741185 0.75 LRRK2 (0.40) PRKACAPRKACGPRKACBLRRK2KDM4E
SCHEMBL31622333 0.75 LRRK2 (0.40) PRKACAPRKACGPRKACBLRRK2KDM4E
SCHEMBL1261198 0.75 NOS2 (0.54) PRKACAPRKACGPRKACBLRRK2NOS3
SCHEMBL22980341 0.75 PRKACA (0.38) PRKACAPRKACGPRKACBLRRK2NOS3
SCHEMBL565899 0.75 HTT (0.41) PRKACAPRKACGPRKACBLRRK2NOS3
SCHEMBL30679309 0.71 PRKACA (0.36) PRKACAPRKACGPRKACBLRRK2NOS3
SCHEMBL564697 0.71 ALDH1A1 (0.53) PRKACAPRKACGPRKACBKDM4EMEN1
SCHEMBL30731660 0.71 KDM4E (0.41) PRKACAPRKACGPRKACBLRRK2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010060589-A1 INDOLE AND BENZOXAZINE DERIVATIVES AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS ORTHO-MCNEIL-JANSSEN PHARMACEUTICALS, INC. (US) 2010-06-03 WO disclosed