SCHEMBL7912753

SCHEMBL7912753

C=Nc1cc(C)cnc1N(C)C

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
NOS2 P35228 1/20 0.36
CCR1 P32246 1/20 0.32
CCR5 P51681 1/20 0.32
CCR8 P51685 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15061923 0.73 NOS3 (0.54) NOS3NOS1NOS2CCR1CCR5
SCHEMBL7922466 0.71 NOS3 (0.38) NOS3NOS1NOS2CCR1CCR5
SCHEMBL24148824 0.71 CHEK1 (0.34)
SCHEMBL26894640 0.69 NOS3 (0.40) NOS3NOS1NOS2CCR1CCR5
SCHEMBL17778679 0.69 NOS3 (0.40) NOS3NOS1NOS2CCR1CCR5
SCHEMBL17703483 0.69 NOS1 (0.40) NOS3NOS1NOS2CCR1CCR5
SCHEMBL15061930 0.69 NOS3 (0.40) NOS3NOS1NOS2CCR1CCR5
SCHEMBL20086563 0.67 NOS3 (0.38) NOS3NOS1NOS2CCR1CCR5
SCHEMBL24226815 0.67 ACHE (0.40) NOS3NOS1NOS2CCR1CCR5
SCHEMBL21710342 0.66 NOS2 (0.32) NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2351743-A1 BICYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-08-03 EP disclosed
WO-2010050445-A1 BICYCLIC COMPOUND 武田薬品工業株式会社 (JP) 2010-05-06 WO disclosed