SCHEMBL7913085

SCHEMBL7913085

Nc1c(Nc2cccc(-c3ncc[nH]3)c2)c(=O)c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCP P55072 1/20 0.46
NISCH Q9Y2I1 2/20 0.43
MTOR P42345 1/20 0.43
ADK P55263 1/20 0.43
CCR3 P51677 1/20 0.36
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
KMT2A Q03164 1/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
BRD4 O60885 1/20 0.34
PARP1 P09874 2/20 0.34
MAPKAPK2 P49137 3/20 0.34
ITGB3 P05106 1/20 0.33
ITGAV P06756 1/20 0.33
HCRTR1 O43613 1/20 0.33
PLK1 P53350 1/20 0.33
MRGPRX4 Q96LA9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7916081 0.79 CNR1 (0.47) BRD4MAPKAPK2PLK1
SCHEMBL1502186 0.77 MEN1 (0.35) MEN1POLBKMT2AMAPKAPK2PLK1
SCHEMBL7913081 0.77 HDAC3 (0.46) MEN1POLBKMT2ABRD4MAPKAPK2
SCHEMBL7913077 0.77 KDM4E (0.57) KDM4EALDH1A1MEN1POLBKMT2A
SCHEMBL7905830 0.76 SIRT2 (0.48) KDM4EALDH1A1MEN1POLBKMT2A
SCHEMBL7905484 0.75 MEN1 (0.50) ALDH1A1MEN1KMT2A
SCHEMBL7905810 0.74 HPGDS (0.38) MEN1POLBKMT2ABRD4MAPKAPK2
SCHEMBL7913791 0.73 CXCR2 (0.37) MTORKDM4EALDH1A1MEN1POLB
SCHEMBL24782866 0.73 NISCH (0.55) VCPNISCHMTORADKCCR3
SCHEMBL7915476 0.73 CNR1 (0.45) MEN1POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211220-B1 ANTITUMOR AGENTS AND ANTICARCIINOGENIC AGENTS CELL PATHWAYS, INC. 2001-04-03 US claimed
US-6211220-B1 ANTITUMOR AGENTS AND ANTICARCIINOGENIC AGENTS CELL PATHWAYS, INC. 2001-04-03 US disclosed
WO-1994029277-A1 AMILINO- OR PYRIDYLAMINO- CYCLOBUTENE- 1,2-DIONE DERIVATIVES AS cGMP PHOSPHODIESTERASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 1994-12-22 WO disclosed