SCHEMBL7905810

SCHEMBL7905810

Nc1c(Nc2cccc(-c3ncco3)c2)c(=O)c1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.38
JAK3 P52333 1/20 0.36
IMPDH2 P12268 1/20 0.36
MAPKAPK2 P49137 3/20 0.36
ABL1 P00519 1/20 0.35
EGFR P00533 1/20 0.35
BCR P11274 1/20 0.35
SRC P12931 1/20 0.35
PRKACA P17612 1/20 0.35
PRKACG P22612 1/20 0.35
PRKACB P22694 1/20 0.35
BRD4 O60885 1/20 0.35
PLK1 P53350 1/20 0.35
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
KMT2A Q03164 1/20 0.35
HDAC4 P56524 3/20 0.34
SYK P43405 3/20 0.34
BACE1 P56817 1/20 0.34
BACE2 Q9Y5Z0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7913081 0.77 HDAC3 (0.46) MAPKAPK2ABL1BCRSRCBRD4
SCHEMBL7916081 0.76 CNR1 (0.47) MAPKAPK2ABL1BCRBRD4PLK1
SCHEMBL7905830 0.76 SIRT2 (0.48) PLK1MEN1POLBKMT2AHDAC3
SCHEMBL4477549 0.75 SYK (0.48) ABL1EGFRBCRSRCPRKACA
SCHEMBL7905484 0.75 MEN1 (0.50) ABL1EGFRBCRSRCPRKACA
SCHEMBL7913085 0.74 VCP (0.46) MAPKAPK2BRD4PLK1MEN1POLB
SCHEMBL7913791 0.73 CXCR2 (0.37) ABL1EGFRBCRSRCPRKACA
SCHEMBL21646502 0.73 HPGDS (0.46) HPGDSJAK3IMPDH2BRD4PLK1
SCHEMBL7915476 0.73 CNR1 (0.45) ABL1EGFRBCRSRCPRKACA
SCHEMBL1502186 0.72 MEN1 (0.35) MAPKAPK2ABL1EGFRBCRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211220-B1 ANTITUMOR AGENTS AND ANTICARCIINOGENIC AGENTS CELL PATHWAYS, INC. 2001-04-03 US claimed
US-6211220-B1 ANTITUMOR AGENTS AND ANTICARCIINOGENIC AGENTS CELL PATHWAYS, INC. 2001-04-03 US disclosed
WO-1994029277-A1 AMILINO- OR PYRIDYLAMINO- CYCLOBUTENE- 1,2-DIONE DERIVATIVES AS cGMP PHOSPHODIESTERASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 1994-12-22 WO disclosed