SCHEMBL7915364

SCHEMBL7915364

Cc1ccc(-c2cnccn2)c(N)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MBOAT4 Q96T53 1/20 0.47
HTT P42858 1/20 0.40
RECQL P46063 1/20 0.40
KDM4E B2RXH2 1/20 0.39
GLA P06280 1/20 0.39
ALOX5AP P20292 2/20 0.39
FEN1 P39748 2/20 0.39
PIK3CD O00329 1/20 0.37
PIK3CA P42336 1/20 0.37
PIK3CB P42338 1/20 0.37
PI4KA P42356 1/20 0.37
PIK3CG P48736 1/20 0.37
PI4KB Q9UBF8 1/20 0.37
HSP90AA1 P07900 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
PIM1 P11309 1/20 0.35
PIM3 Q86V86 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15436237 0.82 PIM1 (0.45) MBOAT4HTTRECQLKDM4EGLA
Hydrochloric Acid SCHEMBL15436253 0.81 PIM1 (0.44) MBOAT4HTTRECQLKDM4EGLA
Hydrochloric Acid SCHEMBL27850418 0.81 PIM1 (0.44) MBOAT4HTTRECQLKDM4EGLA
SCHEMBL7910798 0.77 KDM4E (0.46) HTTKDM4EHSP90AA1ALDH1A1CYP1A2
SCHEMBL3389640 0.76 WNT3A (0.35) MBOAT4HTTRECQLMEN1KMT2A
SCHEMBL2470786 0.74 PIM2 (0.40) KDM4EMEN1KMT2AALDH1A1PIM1
SCHEMBL31372672 0.74 PIM2 (0.40) KDM4EMEN1KMT2AALDH1A1PIM1
SCHEMBL7911485 0.74 CDK2 (0.41) HTTKDM4EGLAALDH1A1ROCK1
SCHEMBL19376940 0.73 ALOX5AP (0.44) MBOAT4ALOX5APFEN1PIK3CDPIK3CA
SCHEMBL15436242 0.73 DHFR (0.46) MBOAT4HTTRECQLKDM4EGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063663-A1 N-{[(IR,4S,6R-3-(2-PYRIDINYLCARBONYL)-3-AZABICYCLO [4.1.0]HEPT-4-YL] METHYL}-2-HETEROARYLAMINE DERIVATIVES AND USES THEREOF GLAXO GROUP LIMITED (GB) 2010-06-10 WO disclosed