SCHEMBL15436237

SCHEMBL15436237

Nc1ccc(-c2cnccn2)c(N)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 2/20 0.45
PIM2 Q9P1W9 2/20 0.45
PIM3 Q86V86 1/20 0.45
MBOAT4 Q96T53 1/20 0.43
HSP90AA1 P07900 1/20 0.43
ALOX5AP P20292 3/20 0.43
FEN1 P39748 3/20 0.43
PIK3CD O00329 1/20 0.39
PIK3CA P42336 1/20 0.39
PIK3CB P42338 1/20 0.39
PI4KA P42356 1/20 0.39
PIK3CG P48736 1/20 0.39
PI4KB Q9UBF8 1/20 0.39
KDM4E B2RXH2 1/20 0.38
GLA P06280 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
PKM P14618 1/20 0.36
METAP2 P50579 1/20 0.36
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL15436253 0.98 PIM1 (0.44) PIM1PIM2PIM3MBOAT4HSP90AA1
Hydrochloric Acid SCHEMBL27850418 0.98 PIM1 (0.44) PIM1PIM2PIM3MBOAT4HSP90AA1
Maleic Acid SCHEMBL28393695 0.87 PIM2 (0.44) PIM1PIM2PIM3MBOAT4HSP90AA1
Maleic Acid SCHEMBL30608269 0.87 PIM2 (0.44) PIM1PIM2PIM3MBOAT4HSP90AA1
SCHEMBL7915364 0.82 MBOAT4 (0.47) PIM1PIM2PIM3MBOAT4HSP90AA1
SCHEMBL901793 0.78 ADORA2B (0.55) PIM1PIM2PIM3MBOAT4HSP90AA1
SCHEMBL15436242 0.76 DHFR (0.46) MBOAT4HSP90AA1ALOX5APFEN1PIK3CD
SCHEMBL798061 0.76 KDM4E (0.50) HSP90AA1PI4KAPI4KBKDM4EGLA
SCHEMBL19376940 0.76 ALOX5AP (0.44) MBOAT4HSP90AA1ALOX5APFEN1PIK3CD
SCHEMBL27960699 0.75 NCF1 (0.45) PIM1PIM2PIM3ALOX5APFEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102307869-B Aminopyrazine derivative and medicine NIPPON SHINYAKU CO.,LTD. (JP) 2014-10-22 CN claimed
CN-102307869-B Aminopyrazine derivative and medicine NIPPON SHINYAKU CO.,LTD. (JP) 2014-10-22 CN disclosed
EP-2394999-B1 AMINOPYRAZINE DERIVATIVE AND MEDICINE NIPPON SHINYAKU CO LTD (JP) 2014-01-29 EP disclosed
CN-102307869-A Aminopyrazine derivative and medicine NIPPON SHINYAKU CO LTD 2012-01-04 CN disclosed
EP-2394999-A1 AMINOPYRAZINE DERIVATIVE AND MEDICINE Nippon Shinyaku Co., Ltd. (JP) 2011-12-14 EP disclosed