SCHEMBL7917047

SCHEMBL7917047

O=C1NCC=NN1c1ccc(C(F)c2ccc(Cl)cc2)c(Cl)c1

nearest known ligand 0.31

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
MEN1 O00255 1/20 0.30
NR1I2 O75469 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7917049 0.87 MEN1 (0.34) MEN1NR1I2KMT2A
SCHEMBL7917708 0.86 CHEK2 (0.35) CYP3A4CYP2D6MEN1NR1I2KMT2A
SCHEMBL7917757 0.83 FPR2 (0.33) MEN1NR1I2KMT2A
SCHEMBL7917733 0.78 MEN1 (0.33) MEN1NR1I2KMT2A
SCHEMBL7917510 0.77 MEN1 (0.34) MEN1NR1I2KMT2A
SCHEMBL7919693 0.77 MEN1 (0.34) CYP3A4MEN1NR1I2KMT2A
SCHEMBL7919222 0.77 CNR1 (0.33)
SCHEMBL7922600 0.77 MEN1 (0.32) CYP2D6MEN1NR1I2KMT2A
SCHEMBL7919716 0.76 SCN8A (0.32)
SCHEMBL7917715 0.76 SCN8A (0.34) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211178-B1 ANTIPROTOZOA AGENTS FOR COCCIDIOIDES; CYCLIZATION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-03 US disclosed
EP-0648760-B1 Triazine derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-01-27 EP disclosed
EP-0648760-A2 Triazine derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-04-19 EP disclosed