SCHEMBL7917708

SCHEMBL7917708

O=C1NCC=NN1c1ccc(C(O)c2ccc(Cl)cc2)c(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.35
TOP2A P11388 1/20 0.33
TOP2B Q02880 1/20 0.33
BRD4 O60885 1/20 0.31
CYP3A4 P08684 2/20 0.31
CYP2D6 P10635 1/20 0.31
ROCK2 O75116 1/20 0.30
DRD4 P21917 3/20 0.30
MEN1 O00255 1/20 0.30
NR1I2 O75469 1/20 0.30
KMT2A Q03164 1/20 0.30
ADRA2C P18825 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7919693 0.87 MEN1 (0.34) CYP3A4ROCK2DRD4MEN1NR1I2
SCHEMBL7917047 0.86 CYP3A4 (0.31) CYP3A4CYP2D6MEN1NR1I2KMT2A
SCHEMBL7990341 0.80 ALDH1A1 (0.33) DRD4
SCHEMBL7917049 0.77 MEN1 (0.34) MEN1NR1I2KMT2A
SCHEMBL7917510 0.77 MEN1 (0.34) MEN1NR1I2KMT2A
SCHEMBL7917015 0.77 DRD4 (0.32) CYP2D6DRD4MEN1NR1I2KMT2A
SCHEMBL7917715 0.76 SCN8A (0.34) CYP3A4
SCHEMBL7910016 0.75 SRD5A2 (0.43) CHEK2MEN1KMT2A
SCHEMBL7917733 0.75 MEN1 (0.33) MEN1NR1I2KMT2A
SCHEMBL7919224 0.75 MEN1 (0.33) CYP2D6DRD4MEN1NR1I2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211178-B1 ANTIPROTOZOA AGENTS FOR COCCIDIOIDES; CYCLIZATION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-03 US disclosed
US-5994355-A ANTIPROTOZOA AGENTS, PARASITICIDE; VETERINARY MEDICINE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-11-30 US disclosed
EP-0648760-B1 Triazine derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-01-27 EP disclosed
EP-0648760-A2 Triazine derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-04-19 EP disclosed