SCHEMBL7918146

SCHEMBL7918146

COc1cc(C(=O)NC(C)(C)C)ccc1S(=O)(=O)n1nc(C(F)(F)F)n(C)c1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.38
TSHR P16473 1/20 0.38
HPGD P15428 1/20 0.38
MAPT P10636 4/20 0.38
POLB P06746 2/20 0.38
ANO1 Q5XXA6 3/20 0.38
AVPR1A P37288 1/20 0.37
PTK2 Q05397 1/20 0.37
LRRK2 Q5S007 1/20 0.36
KMT2A Q03164 3/20 0.36
RAB9A P51151 2/20 0.36
MEN1 O00255 2/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
ALOX12 P18054 1/20 0.36
CYP2C19 P33261 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7911467 0.79 ALDH1A1 (0.39) L3MBTL1HPGDMAPTPOLBAVPR1A
SCHEMBL16167675 0.79 ALDH1A1 (0.39) L3MBTL1TSHRHPGDMAPTANO1
SCHEMBL7908197 0.78 ALDH1A1 (0.38) HPGDMAPTAVPR1APTK2LRRK2
SCHEMBL7914828 0.77 AVPR1A (0.39) TSHRHPGDMAPTAVPR1APTK2
SCHEMBL7909318 0.76 AVPR1A (0.37) L3MBTL1HPGDMAPTAVPR1ALRRK2
SCHEMBL7908194 0.76 KMT2A (0.38) TSHRHPGDMAPTAVPR1APTK2
SCHEMBL16167674 0.75 AVPR1A (0.37) HPGDMAPTPOLBAVPR1APTK2
SCHEMBL2504845 0.74 AVPR2 (0.48) AVPR1A
SCHEMBL7909327 0.74 AVPR1A (0.39) L3MBTL1HPGDMAPTPOLBAVPR1A
SCHEMBL16167673 0.74 HSD11B1 (0.40) L3MBTL1AVPR1AKMT2AALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8859601-B2 Substituted benzyl and phenylsulfonyl triazolones, and use thereof BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-10-14 US disclosed
US-8859601-B2 Substituted benzyl and phenylsulfonyl triazolones, and use thereof BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-10-14 US disclosed
WO-2010063402-A1 SUBSTITUTED BENZYL AND PHENYLSULFONYL TRIAZOLONES, AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-06-10 WO disclosed