SCHEMBL7919781

SCHEMBL7919781

C=C(O)c1ccc2cccc(-c3cccc4ccncc34)c2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNF P01375 3/20 0.54
HIPK2 Q9H2X6 1/20 0.40
HTR2C P28335 2/20 0.39
MAPK10 P53779 2/20 0.38
SLC22A12 Q96S37 2/20 0.37
HDAC6 Q9UBN7 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MAPKAPK2 P49137 1/20 0.36
CYP1A1 P04798 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP1B1 Q16678 1/20 0.35
CSNK2A2 P19784 4/20 0.35
CSNK2B P67870 3/20 0.35
PIK3CD O00329 1/20 0.35
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35
CSNK2A1 P68400 2/20 0.33
PIM1 P11309 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16502698 0.85 TNF (0.54) TNFHIPK2SLC22A12CSNK2A2CSNK2B
SCHEMBL7917731 0.84 TNF (0.49) TNFHIPK2KDM4ECYP1A1CYP1A2
SCHEMBL7916601 0.81 TNF (0.43) TNFHIPK2HTR2CHDAC6KDM4E
SCHEMBL7920176 0.78 CCR1 (0.46) HDAC6KDM4ECYP3A4CYP2D6
SCHEMBL16502680 0.78 CYP19A1 (0.51) TNFHIPK2MAPK10KDM4ECSNK2A2
SCHEMBL7917427 0.77 F2 (0.41) TNFHDAC6KDM4E
SCHEMBL7920129 0.76 TNF (0.45) TNFHDAC6KDM4ECYP1A2
SCHEMBL16502832 0.76 SLC9A1 (0.49) TNFHIPK2HTR2C
SCHEMBL7918345 0.76 CYP1A2 (0.40) KDM4ECYP1A1CYP1A2CYP1B1
SCHEMBL7916817 0.76 AKR1C3 (0.41) HDAC6KDM4ECYP1A1CYP1A2CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010090304-A1 ACYLGUANIDINE DERIVATIVE アステラス製薬株式会社 (JP) 2010-08-12 WO disclosed