SCHEMBL7920089

SCHEMBL7920089

COc1ccccc1-c1cc(=O)n2ccccc2n1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.49
DCTPP1 Q9H773 1/20 0.48
TLR9 Q9NR96 1/20 0.46
MAPT P10636 3/20 0.45
LMNA P02545 2/20 0.45
TP53 P04637 1/20 0.45
KDM4E B2RXH2 3/20 0.45
HSD17B10 Q99714 1/20 0.45
HSP90AB1 P08238 1/20 0.45
RXFP1 Q9HBX9 2/20 0.44
HPGD P15428 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
ALDH1A1 P00352 1/20 0.44
POLB P06746 1/20 0.44
GAA P10253 1/20 0.44
ADORA3 P0DMS8 3/20 0.43
ADORA1 P30542 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7920470 0.85 KDM4E (0.54) HSP90AA1DCTPP1MAPTTP53KDM4E
SCHEMBL32688343 0.83 DCTPP1 (0.48) HSP90AA1DCTPP1MAPTLMNATP53
SCHEMBL7920187 0.83 DCTPP1 (0.48) HSP90AA1DCTPP1MAPTLMNATP53
SCHEMBL890511 0.81 DPP4 (0.49) HSP90AA1MAPTTP53KDM4EHSP90AB1
SCHEMBL10690765 0.81 KDM4E (0.61) MAPTTP53KDM4EHSD17B10HPGD
SCHEMBL7920397 0.78 HSP90AA1 (0.50) HSP90AA1DCTPP1MAPTLMNATP53
SCHEMBL8108255 0.78 KDM4E (0.65) MAPTTP53KDM4EHSD17B10KMT2A
SCHEMBL8102203 0.77 HSP90AA1 (0.47) HSP90AA1MAPTKDM4EHSP90AB1HPGD
SCHEMBL30433019 0.76 KDM4E (0.61) MAPTKDM4EHSD17B10HPGDKMT2A
SCHEMBL7925220 0.76 MEN1 (0.57) MAPTLMNATP53KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6229016-B1 PYRIDOPYRIMIDINE DERIVATIVES AS CHEMICAL INTERMEDIATES; POLYMERIZATION INHIBITION OF TUBULIN THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL 2001-05-08 US disclosed
US-6071930-A FOR INHIBITION OF MITOSIS OR TUMOR GROWTH THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2000-06-06 US disclosed
US-5994367-A PREVENT CELL MITOSIS; ANTICARCINOGENIC AGENTS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1999-11-30 US disclosed