SCHEMBL7920105

SCHEMBL7920105

COc1cccc(-c2cc(=O)n3cc(Cl)ccc3n2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A3 P47895 3/20 0.59
ALDH1A1 P00352 4/20 0.51
HPGD P15428 4/20 0.51
KDM4E B2RXH2 3/20 0.51
RAB9A P51151 3/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
NPC1 O15118 2/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
LMNA P02545 1/20 0.48
PKM P14618 1/20 0.48
NFKB1 P19838 1/20 0.48
STAT3 P40763 1/20 0.48
STAT1 P42224 1/20 0.48
NFKB2 Q00653 1/20 0.48
RELA Q04206 1/20 0.48
WDR5 P61964 1/20 0.44
BRD4 O60885 1/20 0.44
SLC2A1 P11166 1/20 0.44
TLR8 Q9NR97 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8099894 0.86 MEN1 (0.52) ALDH1A3ALDH1A1HPGDKDM4ERAB9A
SCHEMBL7925168 0.85 MEN1 (0.51) ALDH1A3ALDH1A1HPGDKDM4ERAB9A
SCHEMBL28958142 0.82 NPC1 (0.56) ALDH1A3ALDH1A1HPGDKDM4ERAB9A
SCHEMBL7925220 0.81 MEN1 (0.57) ALDH1A3ALDH1A1HPGDKDM4ERAB9A
SCHEMBL8106156 0.80 PKM (0.45) ALDH1A3ALDH1A1HPGDKDM4ERAB9A
SCHEMBL13325709 0.80 ALDH1A3 (0.83) ALDH1A3ALDH1A1HPGDKDM4ERAB9A
SCHEMBL21902775 0.80 MEN1 (0.55) ALDH1A3ALDH1A1MEN1KMT2ALMNA
SCHEMBL15174027 0.79 ALDH1A1 (0.50) ALDH1A3ALDH1A1HPGDKDM4ERAB9A
SCHEMBL15173858 0.78 ADRB1 (0.51) MEN1KMT2AWDR5CLK4TSHR
SCHEMBL1658718 0.78 MEN1 (0.46) ALDH1A3MEN1KMT2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6229016-B1 PYRIDOPYRIMIDINE DERIVATIVES AS CHEMICAL INTERMEDIATES; POLYMERIZATION INHIBITION OF TUBULIN THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL 2001-05-08 US disclosed
US-6071930-A FOR INHIBITION OF MITOSIS OR TUMOR GROWTH THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2000-06-06 US disclosed
US-5994367-A PREVENT CELL MITOSIS; ANTICARCINOGENIC AGENTS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1999-11-30 US disclosed