SCHEMBL7920760

SCHEMBL7920760

C1=C(c2c[nH]c3ncccc23)CCN(CC2CN(c3ccccc3)c3ccccc3O2)C1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 1/20 0.55
SIGMAR1 Q99720 1/20 0.55
HTR1A P08908 12/20 0.53
SLC6A4 P31645 5/20 0.50
DRD2 P14416 3/20 0.47
DRD4 P21917 3/20 0.47
DRD3 P35462 2/20 0.47
ADRA1D P25100 1/20 0.46
ADRA1A P35348 1/20 0.46
ADRA1B P35368 1/20 0.46
CHEK1 O14757 2/20 0.44
MAP4K4 O95819 2/20 0.44
PIM1 P11309 2/20 0.44
PRKACA P17612 2/20 0.44
CLK2 P49760 2/20 0.44
GSK3B P49841 2/20 0.44
CDK5 Q00535 2/20 0.44
PRKAA1 Q13131 2/20 0.44
ROCK1 Q13464 2/20 0.44
DYRK1A Q13627 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5844134 0.74 HTR1A (0.61) TMEM97SIGMAR1HTR1ASLC6A4ADRA1D
SCHEMBL13502652 0.73 SIGMAR1 (0.68) TMEM97SIGMAR1HTR1ASLC6A4DRD2
SCHEMBL6108012 0.71 HTR1A (0.65) TMEM97SIGMAR1HTR1ASLC6A4DRD2
SCHEMBL9529716 0.71 KCNH2 (0.50) HTR1ADRD2DRD4ADRA1DADRA1A
Hydrochloric Acid SCHEMBL10368330 0.71 ABCB1 (0.48) SIGMAR1HTR1ADRD2DRD4DRD3
SCHEMBL13064304 0.70 TMEM97 (0.59) TMEM97SIGMAR1HTR1ASLC6A4DRD2
SCHEMBL9530044 0.69 ABCB1 (0.49) SIGMAR1HTR1ADRD2DRD4DRD3
SCHEMBL9696810 0.69 ADRA2A (0.59) SIGMAR1HTR1AADRA1DADRA1AADRA1B
SCHEMBL7911460 0.69 HTR1A (1.00) SIGMAR1HTR1ASLC6A4DRD2HTR2A
SCHEMBL9455117 0.69 CASR (0.45) TMEM97SIGMAR1HTR1ADRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6221863-B1 TREATING DEPRESSION IN A PATIENT AMERICAN HOME PRODUCTS CORP. 2001-04-24 US disclosed
WO-2000040581-A1 3,4-DIHYDRO-2H-BENZO[1,4]OXAZINE DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 2000-07-13 WO disclosed