SCHEMBL7922222

SCHEMBL7922222

Cc1nc(C2(C(=O)O)C=CC(c3ccccc3C)C=C2)no1

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 2/20 0.34
P2RX3 P56373 13/20 0.32
ADORA2A P29274 3/20 0.32
ADORA1 P30542 1/20 0.32
PLK1 P53350 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7922191 0.69 ADORA2A (0.30) P2RX3ADORA2AADORA1
SCHEMBL7922225 0.65 NR1H4 (0.39) NR1H4
SCHEMBL17393757 0.63 ACHE (0.47)
SCHEMBL7913508 0.62 ADORA2A (0.38) ADORA2AADORA1PLK1
SCHEMBL20566162 0.61 HTR2C (0.35)
SCHEMBL7219943 0.59 HDAC4 (0.36)
SCHEMBL9849476 0.58 TSHR (0.45)
SCHEMBL12660084 0.57 NPC1 (0.62) NR1H4
SCHEMBL4075982 0.57 HDAC4 (0.37) NR1H4
SCHEMBL1281643 0.57 NPC1 (0.64) NR1H4PLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001766-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2001-04-04 EP disclosed
EP-1001766-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2000-05-24 EP disclosed
WO-1999001127-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 1999-01-14 WO disclosed