SCHEMBL7922538

SCHEMBL7922538

CN1C(=O)CNN(c2cc(Cl)cc(Cl)c2)C1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.35
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
ADRB1 P08588 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
BCL2A1 Q16548 1/20 0.33
ALDH1A1 P00352 3/20 0.32
RECQL P46063 1/20 0.32
DRD2 P14416 1/20 0.32
DRD3 P35462 1/20 0.32
USP2 O75604 1/20 0.31
BRPF1 P55201 1/20 0.31
ITGB2 P05107 1/20 0.31
ICAM1 P05362 1/20 0.31
ITGAL P20701 1/20 0.31
GAA P10253 1/20 0.31
POLB P06746 1/20 0.31
HPGD P15428 1/20 0.31
OPRK1 P41145 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9823375 0.75 MEN1 (0.49) ALDH1A1GAAPOLBHPGDMEN1
SCHEMBL7919150 0.69 TSHR (0.38) TSHRCHRM2CHRM4ADRB1CHRM1
SCHEMBL8581414 0.68 ESR1 (0.41) BRPF1
SCHEMBL11081029 0.66 ALOX12 (0.47) TSHRALDH1A1DRD2DRD3POLB
SCHEMBL4623495 0.64 HTR3E (0.41) ADRB1ALDH1A1DRD2DRD3POLB
SCHEMBL3838027 0.62 ALDH1A1 (0.47) TSHRBCL2A1ALDH1A1RECQLDRD2
SCHEMBL3841672 0.61 AR (0.50) TSHRCHRM2CHRM4ADRB1CHRM1
SCHEMBL11278830 0.60 TSHR (0.43) TSHRCHRM2CHRM4ADRB1CHRM1
SCHEMBL10268369 0.58 ALDH1A1 (0.50) TSHRCHRM2CHRM4ADRB1CHRM1
Dimethachlon SCHEMBL410360 0.58 TSHR (0.50) TSHRCHRM2CHRM4ADRB1CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211178-B1 ANTIPROTOZOA AGENTS FOR COCCIDIOIDES; CYCLIZATION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-03 US disclosed
US-5994355-A ANTIPROTOZOA AGENTS, PARASITICIDE; VETERINARY MEDICINE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-11-30 US disclosed
EP-0648760-B1 Triazine derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-01-27 EP disclosed
EP-0648760-A2 Triazine derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-04-19 EP disclosed