SCHEMBL7922651

SCHEMBL7922651

NC=S.O=C(Cn1nnc(-c2cccc(C(F)(F)F)c2)n1)NNc1ccc(C(F)(F)F)cc1

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.59
POLB P06746 3/20 0.54
HTT P42858 1/20 0.54
MAPT P10636 3/20 0.53
KDM4E B2RXH2 1/20 0.53
MAPK1 P28482 1/20 0.53
BLM P54132 1/20 0.53
TSHR P16473 1/20 0.53
LMNA P02545 2/20 0.52
XPO1 O14980 1/20 0.52
KMT2A Q03164 2/20 0.50
MEN1 O00255 1/20 0.50
KCNJ6 P48051 1/20 0.50
KCNJ5 P48544 1/20 0.50
KCNJ3 P48549 1/20 0.50
TP53 P04637 3/20 0.48
THRB P10828 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
NTRK1 P04629 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7922641 0.85 MAPT (0.61) ALDH1A1POLBHTTMAPTKDM4E
SCHEMBL27632153 0.79 ALDH1A1 (0.62) ALDH1A1POLBHTTMAPTKDM4E
SCHEMBL3282363 0.78 ALDH1A1 (0.64) ALDH1A1POLBHTTMAPTKDM4E
SCHEMBL14096405 0.75 ALDH1A1 (0.64) ALDH1A1POLBHTTMAPTKDM4E
SCHEMBL14096380 0.75 ALDH1A1 (0.53) ALDH1A1POLBHTTMAPTKDM4E
SCHEMBL7920537 0.70 MAPT (0.46) ALDH1A1POLBHTTMAPTKDM4E
SCHEMBL7922254 0.69 ALDH1A1 (0.44) ALDH1A1POLBHTTMAPTKDM4E
SCHEMBL16126203 0.68 XPO1 (1.00) ALDH1A1POLBHTTMAPTTSHR
SCHEMBL7922259 0.68 TASP1 (0.61) ALDH1A1POLBMAPTKDM4EMAPK1
SCHEMBL7829737 0.67 ALDH1A1 (0.73) ALDH1A1POLBHTTMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100500-A1 THE USE OF CD4-BINDING SMALL MOLECULES TO INHIBIT HIV INFECTION THOMAS JEFFERSON UNIVERSITY (US) 2001-05-23 EP claimed
WO-2000004903-A1 THE USE OF CD4-BINDING SMALL MOLECULES TO INHIBIT HIV INFECTION THOMAS JEFFERSON UNIVERSITY (US) 2000-02-03 WO claimed