SCHEMBL7926845

SCHEMBL7926845

NC(=O)c1cc[nH]c1C(N)=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 2/20 0.47
IKBKB O14920 6/20 0.40
CHUK O15111 5/20 0.40
ALDH1A1 P00352 3/20 0.39
ATM Q13315 1/20 0.39
GDA Q9Y2T3 1/20 0.39
MAPT P10636 2/20 0.38
KDM4E B2RXH2 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CSNK1A1 P48729 1/20 0.38
TYRO3 Q06418 1/20 0.38
DYRK1B Q9Y463 1/20 0.38
BTK Q06187 1/20 0.38
NUDT1 P36639 1/20 0.37
PARP1 P09874 1/20 0.36
MEN1 O00255 1/20 0.35
MAPK1 P28482 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5653478 0.86 KEAP1 (0.41) PDPK1IKBKBCHUKALDH1A1ATM
SCHEMBL29158222 0.85 CSNK1A1 (0.40) PDPK1IKBKBCHUKALDH1A1ATM
SCHEMBL4783577 0.78
SCHEMBL562266 0.76
SCHEMBL162641 0.76
SCHEMBL6672416 0.76
SCHEMBL30884200 0.76 PDPK1 (0.43) PDPK1IKBKBCHUKALDH1A1ATM
SCHEMBL5609871 0.76 PDPK1 (0.43) PDPK1IKBKBCHUKALDH1A1ATM
SCHEMBL16043412 0.74
SCHEMBL849718 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-120192278-A Azole bisamide-containing compound and preparation method and application thereof 江西天宇化工有限公司 2025-06-24 CN claimed
CN-120192278-A Azole bisamide-containing compound and preparation method and application thereof 江西天宇化工有限公司 2025-06-24 CN disclosed
CN-120192278-A Azole bisamide-containing compound and preparation method and application thereof 江西天宇化工有限公司 2025-06-24 CN disclosed
CN-120192278-A Azole bisamide-containing compound and preparation method and application thereof 江西天宇化工有限公司 2025-06-24 CN disclosed
US-9884860-B2 Fused pyrroledicarboxamides and their use as pharmaceuticals SANOFI (FR) 2018-02-06 US disclosed
US-9884860-B2 Fused pyrroledicarboxamides and their use as pharmaceuticals SANOFI (FR) 2018-02-06 US disclosed
US-9884860-B2 Fused pyrroledicarboxamides and their use as pharmaceuticals SANOFI (FR) 2018-02-06 US disclosed
EP-2809669-B1 FUSED PYRROLEDICARBOXAMIDES AND THEIR USE AS PHARMACEUTICALS SANOFI SA (FR) 2017-02-01 EP disclosed
US-20160159793-A1 Fused Pyrroledicarboxamides and Their Use as Pharmaceuticals SANOFI (FR) 2016-06-09 US disclosed
US-20160159793-A1 Fused Pyrroledicarboxamides and Their Use as Pharmaceuticals SANOFI (FR) 2016-06-09 US disclosed
US-9284333-B2 Fused pyrroledicarboxamides and their use as pharmaceuticals SANOFI (FR) 2016-03-15 US disclosed
EP-2809669-A1 FUSED PYRROLEDICARBOXAMIDES AND THEIR USE AS PHARMACEUTICALS SANOFI (FR) 2014-12-10 EP disclosed
EP-2809669-A1 FUSED PYRROLEDICARBOXAMIDES AND THEIR USE AS PHARMACEUTICALS SANOFI (FR) 2014-12-10 EP disclosed
CN-104169281-A Fused pyrroledicarboxamides and their use as pharmaceuticals SANOFI SA 2014-11-26 CN disclosed
CN-104169281-A Fused pyrroledicarboxamides and their use as pharmaceuticals SANOFI SA 2014-11-26 CN disclosed
WO-2013113860-A1 FUSED PYRROLEDICARBOXAMIDES AND THEIR USE AS PHARMACEUTICALS SANOFI (FR) 2013-08-08 WO disclosed
WO-2013113860-A1 FUSED PYRROLEDICARBOXAMIDES AND THEIR USE AS PHARMACEUTICALS SANOFI (FR) 2013-08-08 WO disclosed
US-6239159-B1 SUBSTRATES FOR POLYMERASE AND TERMINAL TRANSFERASE ENZYMES. CAPABLE OF BASE-PAIRING WITH A NUCLEOTIDE RESIDUE IN A COMPLEMENTARY CHAIN OR BASE STACKING IN THE APPROPRIATE NUCLEIC ACID CHAIN, ADVANTAGE OVER CONVENTIONAL HAPTEN AMERSHAM PHARMACIA BIOTECH UK LIMITED (GB) 2001-05-29 US disclosed
EP-0885235-A1 NUCLEOSIDE ANALOGUES Amersham Pharmacia Biotech UK Limited (GB) 1998-12-23 EP disclosed
WO-1997028176-A1 NUCLEOSIDE ANALOGUES AMERSHAM PHARMACIA BIOTECH UK LIMITED (GB) 1997-08-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160159793-A1 Fused Pyrroledicarboxamides and Their Use as Pharmaceuticals KCNA1, KCNE1, KCNH1 PDPK1 1890/4885IKBKB 4441/4885CHUK 3243/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.