SCHEMBL7928076

SCHEMBL7928076

Cc1csc(NC(=O)c2cc(-c3cccc(Cl)c3)c3nc(C)nn3c2)n1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GCK P35557 4/20 0.60
GRM5 P41594 1/20 0.60
SCD O00767 1/20 0.50
NPC1 O15118 5/20 0.48
RAB9A P51151 5/20 0.48
SMN1; SMN2 Q16637 4/20 0.48
MAPT P10636 4/20 0.48
MEN1 O00255 2/20 0.48
LMNA P02545 2/20 0.48
KMT2A Q03164 2/20 0.48
HPGD P15428 2/20 0.45
ABL1 P00519 1/20 0.44
ALOX12 P18054 1/20 0.44
HTT P42858 1/20 0.44
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7929316 0.85 GCK (0.62) GCKGRM5SCDNPC1RAB9A
SCHEMBL7929315 0.82 SMN1; SMN2 (0.46) GRM5SMN1; SMN2MEN1KMT2AABL1
SCHEMBL7934021 0.80 NPC1 (0.49) GRM5NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL7930891 0.80 POLB (0.50) NPC1RAB9AMAPTMEN1LMNA
SCHEMBL7932092 0.78 KCNQ3 (0.45)
SCHEMBL7934176 0.78 CA2 (0.50) MAPTMEN1LMNAKMT2AKDM4E
SCHEMBL7934179 0.74 DYRK3 (0.50) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL13500910 0.69 CYBB (0.59) GCKGRM5NPC1RAB9ASMN1; SMN2
SCHEMBL7931544 0.69 CNR2 (0.50) GRM5NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL30831954 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059836-A1 SUBSTITUTED AZA-BRIDGED BICYCLICS FOR CARDIOVASCULAR AND CNS DISEASE DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed