Benzenesulfonamide

Benzenesulfonamide

SCHEMBL7929456

N#Cc1cc(-c2ccc(F)cc2)n(-c2ccccc2S(N)(=O)=O)n1.NS(=O)(=O)c1ccccc1

nearest known ligand 0.68

Full drug profile on Sugi Atlas →

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.68
PTGS1 P23219 6/20 0.45
PDPK1 O15530 1/20 0.42
CHRNA7 P36544 2/20 0.41
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8693252 0.95 PTGS2 (0.65) PTGS2PTGS1PDPK1CHRNA7CA1
SCHEMBL8691511 0.88 PTGS2 (0.51) PTGS2PTGS1PDPK1CA1CA2
SCHEMBL8640732 0.84 PTGS2 (0.50) PTGS2PTGS1PDPK1CHRNA7CA2
SCHEMBL8689658 0.84 PTGS2 (0.50) PTGS2PTGS1PDPK1CA1CA2
SCHEMBL8637414 0.84 PTGS2 (0.50) PTGS2PTGS1CA1CA2CA9
SCHEMBL8689144 0.82 PTGS2 (0.48) PTGS2PTGS1CHRNA7CA1CA2
SCHEMBL215235 0.81 PTGS2 (1.00) PTGS2PTGS1CHRNA7CA1CA2
Benzenesulfonamide SCHEMBL7868738 0.80 PTGS2 (0.60) PTGS2PTGS1PDPK1CHRNA7CA1
SCHEMBL8639776 0.80 PTGS2 (0.49) PTGS2PTGS1PDPK1CA1CA2
Sulfamide SCHEMBL7144379 0.80 PTGS2 (0.76) PTGS2PTGS1PDPK1CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2001527542-A 2001-12-25 JP claimed
EP-0979077-A1 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS IN THE PREVENTION OF CARDIOVASCULAR DISORDERS G.D. Searle & Co. (US) 2000-02-16 EP claimed
WO-1998047509-A1 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS IN THE PREVENTION OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1998-10-29 WO claimed