SCHEMBL7929631

SCHEMBL7929631

CCOCCCc1ccc(OB(Oc2ccc(CCCOCC)cc2)Oc2ccc(CCCOCC)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.39
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 1/20 0.39
USP2 O75604 1/20 0.39
LMNA P02545 1/20 0.39
CYP3A4 P08684 1/20 0.39
MAPK1 P28482 1/20 0.39
CASP1 P29466 1/20 0.39
KMT2A Q03164 1/20 0.39
SLCO1B3 Q9NPD5 1/20 0.39
SLCO1B1 Q9Y6L6 1/20 0.39
KDM4E B2RXH2 3/20 0.38
THRB P10828 1/20 0.38
RAB9A P51151 1/20 0.38
CALM1 P0DP23 1/20 0.37
KCNH2 Q12809 1/20 0.36
HPGD P15428 2/20 0.36
HRH3 Q9Y5N1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7216080 0.86 SMN1; SMN2 (0.40) TDP1L3MBTL1SMN1; SMN2ALDH1A1MEN1
SCHEMBL6352411 0.81 ALDH1A1 (0.43) SMN1; SMN2ALDH1A1LMNACYP3A4KDM4E
SCHEMBL2773644 0.81 CA2 (0.52) L3MBTL1SMN1; SMN2ALDH1A1MEN1USP2
SCHEMBL7928439 0.80 TDP1 (0.37) TDP1L3MBTL1SMN1; SMN2LMNAKDM4E
SCHEMBL1487719 0.79 LPL (0.53) SMN1; SMN2ALDH1A1MEN1USP2LMNA
SCHEMBL2769520 0.78 ESR1 (0.55) SMN1; SMN2ALDH1A1MEN1USP2LMNA
SCHEMBL2770828 0.78 ESR1 (0.55) SMN1; SMN2ALDH1A1MEN1USP2LMNA
SCHEMBL718156 0.78 ESR1 (0.55) SMN1; SMN2ALDH1A1MEN1USP2LMNA
SCHEMBL20419190 0.77 POLB (0.45) TDP1L3MBTL1SMN1; SMN2ALDH1A1MEN1
SCHEMBL7928359 0.77 IDO1 (0.36) TDP1L3MBTL1SMN1; SMN2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140896-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 Takeda Chemical Industries, Ltd. (JP) 2001-10-10 EP disclosed
US-6235771-B1 AIDS THERPAY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
WO-2000037455-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-06-29 WO disclosed