SCHEMBL7931301

SCHEMBL7931301

BrCc1ccc2ccccc2c1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HSD17B10 Q99714 2/20 0.41
CYP2A6 P11509 1/20 0.41
TSHR P16473 1/20 0.41
WDR5 P61964 1/20 0.40
GABRA1 P14867 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
HPRT1 P00492 1/20 0.38
MAPT P10636 3/20 0.37
ESR1 P03372 2/20 0.37
ESR2 Q92731 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPK1 P28482 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
NPC1 O15118 1/20 0.36
LMNA P02545 1/20 0.36
RECQL P46063 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30066580 0.88 ALDH1A1 (0.48) TDP1ALDH1A1HSD17B10CYP2A6TSHR
SCHEMBL5691676 0.88 ALDH1A1 (0.48) TDP1ALDH1A1HSD17B10CYP2A6TSHR
SCHEMBL7607961 0.85 MAPT (0.39) TDP1ALDH1A1HSD17B10CYP2A6TSHR
SCHEMBL7604074 0.82 WDR5 (0.46) TDP1ALDH1A1HSD17B10CYP2A6TSHR
SCHEMBL1930924 0.81 ALDH1A1 (0.43) TDP1ALDH1A1TSHRMAPTESR1
SCHEMBL7600324 0.81 WDR5 (0.44) TDP1ALDH1A1HSD17B10CYP2A6TSHR
SCHEMBL6681906 0.81 HPGDS (0.45) TDP1ALDH1A1HSD17B10CYP2A6TSHR
SCHEMBL5240843 0.79 DNMT1 (0.42) TDP1ALDH1A1HSD17B10CYP2A6TSHR
Phosphine SCHEMBL28241012 0.79 HPGDS (0.44) TDP1ALDH1A1HSD17B10CYP2A6TSHR
SCHEMBL17360625 0.79 GPR55 (0.46) GABRA1GABRG2GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1123938-A2 Organometallic fluorenyl compounds, preparation, and use PHILLIPS PETROLEUM COMPANY (US) 2001-08-16 EP disclosed
US-5604242-A ALKOXY- AND CARBOXY-SUBSTITUTED PIPERIDINES FOR SUPPRESSING UPTAKE OF GAMMA-AMINOBUTYRIC ACID, ANALGESICS, ANXIOLYTIC OR ANTIEPILEPTIC AGENTS NOVO NORDISK A/S (DK) 1997-02-18 US disclosed
CN-1128989-A N-substituted azaheterocylic carboxylic acid and esters thereof NOVO NORDISK AS (DK) 1996-08-14 CN disclosed
EP-0705248-A1 N-SUBSTITUTED AZAHETEROCYCLIC CARBOXYLIC ACIDS AND ESTERS THEREOF NOVO NORDISK A/S (DK) 1996-04-10 EP disclosed
EP-0672675-A1 Organometallic fluorenyl compounds, preparation, and use PHILLIPS PETROLEUM COMPANY (US) 1995-09-20 EP disclosed
US-5451649-A Organometallic fluorenyl compounds, preparation, and use PHILLIPS PETROLEUM COMPANY (US) 1995-09-19 US disclosed
WO-1995000486-A1 N-SUBSTITUTED AZAHETEROCYCLIC CARBOXYLIC ACIDS AND ESTERS THEREOF NOVO NORDISK A/S (DK) 1995-01-05 WO disclosed