Bromide

Bromide

SCHEMBL7931348

Br.COc1cc(Br)ccc1N

nearest known ligand 0.59

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADRA2B known ✓ P18089 1/20 0.46
ALDH1A1 P00352 5/20 0.59
CYP3A4 P08684 3/20 0.59
TDP1 Q9NUW8 3/20 0.59
TSHR P16473 1/20 0.59
HSD17B10 Q99714 1/20 0.59
APP P05067 3/20 0.56
POLB P06746 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
MAPT P10636 1/20 0.51
HTT P42858 1/20 0.48
PTGS1 P23219 1/20 0.46
GAA P10253 3/20 0.44
MGAM O43451 1/20 0.44
SI P14410 1/20 0.44
MGAM2 Q2M2H8 1/20 0.44
SLC2A1 P11166 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL155113 0.98 ALDH1A1 (0.61) ALDH1A1CYP3A4TDP1TSHRHSD17B10
Hydrochloric Acid SCHEMBL28039298 0.96 ALDH1A1 (0.61) ALDH1A1CYP3A4TDP1TSHRHSD17B10
SCHEMBL30184653 0.83 ALDH1A1 (0.46) ALDH1A1CYP3A4TDP1TSHRHSD17B10
SCHEMBL29689196 0.80 ALDH1A1 (0.59) ALDH1A1CYP3A4TDP1TSHRHSD17B10
SCHEMBL111151 0.80 ALDH1A1 (0.59) ALDH1A1CYP3A4TDP1TSHRHSD17B10
SCHEMBL1299012 0.79 ALDH1A1 (0.52) ALDH1A1CYP3A4TDP1TSHRHSD17B10
SCHEMBL205027 0.78 GAA (0.47) ALDH1A1CYP3A4TDP1TSHRHSD17B10
SCHEMBL20509 0.77 CA2 (0.56) ALDH1A1CYP3A4TDP1TSHRAPP
SCHEMBL29419589 0.77 CA2 (0.56) ALDH1A1CYP3A4TDP1TSHRAPP
SCHEMBL25033177 0.76 ALDH1A1 (0.43) ALDH1A1CYP3A4TDP1TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235871-B1 Synthesis of oligoarylamines, and uses and reagents related thereto MASSACHUSETTS INSTITUTE OF TECHNOLOGY 2001-05-22 US disclosed
WO-1999028290-A1 SYNTHESIS OF OLIGOARYLAMINES, AND USES AND REAGENTS RELATED THERETO MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1999-06-10 WO disclosed