SCHEMBL7943019

SCHEMBL7943019

NC1=NC2(CCN(C(=O)c3ccc(Br)cc3)CC2)Nc2ccccc21

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NEK2 P51955 1/20 0.59
NOS2 P35228 8/20 0.56
NOS1 P29475 7/20 0.56
ABL1 P00519 3/20 0.47
BCR P11274 3/20 0.47
HPGD P15428 1/20 0.44
NOS3 P29474 2/20 0.43
CA12 O43570 2/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA7 P43166 2/20 0.42
CA9 Q16790 2/20 0.42
CA14 Q9ULX7 2/20 0.42
KCNH2 Q12809 1/20 0.41
KMT2A Q03164 1/20 0.41
SCN5A Q14524 1/20 0.39
SCN9A Q15858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8376992 0.99 NEK2 (0.58) NEK2NOS2NOS1ABL1BCR
SCHEMBL7796711 0.91 NOS2 (0.58) NEK2NOS2NOS1NOS3CA12
SCHEMBL7804452 0.91 NOS2 (0.57) NEK2NOS2NOS1HPGDNOS3
Hydrochloric Acid SCHEMBL8379932 0.90 NOS2 (0.57) NEK2NOS2NOS1NOS3CA12
SCHEMBL7931778 0.90 NOS2 (0.57) NEK2NOS2NOS1NOS3KCNH2
SCHEMBL7796668 0.90 NOS2 (0.57) NEK2NOS2NOS1NOS3CA12
Hydrochloric Acid SCHEMBL8378262 0.90 NOS2 (0.56) NEK2NOS2NOS1HPGDNOS3
Hydrochloric Acid SCHEMBL8377866 0.89 NOS2 (0.56) NEK2NOS2NOS1NOS3CA12
Hydrochloric Acid SCHEMBL8376965 0.89 NOS2 (0.56) NEK2NOS2NOS1NOS3KCNH2
SCHEMBL7805028 0.89 NOS2 (0.56) NEK2NOS2NOS1ABL1BCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6248745-B1 MIXTURE COMPRISING A CYCLOOXYGENASE-2 (COX-2) INHIBITOR AND A 1,2-DIHYDRO-4-AMINOQUINAZOLINE DERIVATIVE INHIBITOR OF INDUCED NITRIC OXIDE SYNTHASE (INOS); NON-STEROIDAL ANTIINFLAMMATORY AGENTS ASTRAZENECA AB (SE) 2001-06-19 US claimed