SCHEMBL7933394

SCHEMBL7933394

C/C=C(\C(=O)O)c1ccc(Cl)cc1F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 4/20 0.45
CYP11B1 P15538 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.43
TSHR P16473 1/20 0.43
CASP1 P29466 1/20 0.43
CXCL12 P48061 1/20 0.42
PPARG P37231 2/20 0.41
PPARA Q07869 2/20 0.41
ALDH1A1 P00352 3/20 0.41
HTT P42858 1/20 0.41
GPR27 Q9NS67 1/20 0.39
GRIK1 P39086 1/20 0.39
ERCC5 P28715 1/20 0.39
FEN1 P39748 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TP53 P04637 1/20 0.39
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
MYC P01106 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7933393 0.84 CXCL12 (0.44) CYP11B2CYP11B1SMN1; SMN2TSHRCASP1
SCHEMBL11093809 0.82 TSHR (0.60) SMN1; SMN2TSHRCASP1ALDH1A1ERCC5
SCHEMBL7942223 0.82 CES2 (0.57) CYP11B2CYP11B1ALDH1A1HTTKMT2A
SCHEMBL7944697 0.82 TSHR (0.60) SMN1; SMN2TSHRCASP1ALDH1A1ERCC5
SCHEMBL7840274 0.78 CES2 (0.50) CYP11B2CYP11B1SMN1; SMN2TSHRCASP1
SCHEMBL9190390 0.78 ERN1 (0.49) SMN1; SMN2TSHRCASP1ALDH1A1ERCC5
SCHEMBL392840 0.77 SMN1; SMN2 (0.63) CYP11B2SMN1; SMN2TSHRCASP1ALDH1A1
SCHEMBL29392929 0.76 MAOB (0.58) CYP11B2CYP11B1SMN1; SMN2TSHRCASP1
SCHEMBL325429 0.76 MAOB (0.58) CYP11B2CYP11B1SMN1; SMN2TSHRCASP1
SCHEMBL27442149 0.75 SMN1; SMN2 (0.48) CYP11B2CYP11B1SMN1; SMN2TSHRCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242634-B1 OF HERBICIDES, HALOPHENYL COMPOUNDS SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2001-06-05 US disclosed
US-6100257-A 2-HALOALKYL,3-(HALOALKYL, ALKENYL, OR ALKYNYL),5-(SUBSTITUTED PHENYL OR HETEROCYCLE),6-ALKYL-PYRIMIDIN-4-ONE COMPOUNDS OF GIVEN STRUCTURE; USE AS HERBICIDES SUMITOMO CHEMICAL COMPANY, LTD. (JP) 2000-08-08 US disclosed
EP-0850229-A1 PYRIMIDIN-4-ONE DERIVATIVES, THEIR USE AS HERBICIDES, INTERMEDIATES FOR THEIR PRODUCTION AND PROCESSES FOR PRODUCING THESE COMPOUNDS SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1998-07-01 EP disclosed
WO-1997006150-A1 PYRIMIDIN-4-ONE DERIVATIVES, THEIR USE AS HERBICIDES, INTERMEDIATES FOR THEIR PRODUCTION AND PROCESSES FOR PRODUCING THESE COMPOUNDS SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-02-20 WO disclosed