SCHEMBL7934084

SCHEMBL7934084

CSCCOc1ccc(OB(Oc2ccc(OCCSC)cc2)Oc2ccc(OCCSC)cc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 8/20 0.39
RAB9A P51151 8/20 0.39
SMN1; SMN2 Q16637 5/20 0.39
HPGD P15428 3/20 0.39
MAPT P10636 3/20 0.39
MAPK1 P28482 2/20 0.39
TP53 P04637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
L3MBTL1 Q9Y468 3/20 0.35
ALDH1A1 P00352 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NQO1 P15559 1/20 0.34
HSD17B10 Q99714 1/20 0.34
LMNA P02545 2/20 0.33
LTA4H P09960 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6343489 0.85 NPC1 (0.37) NPC1RAB9ASMN1; SMN2HPGDMAPT
SCHEMBL13461862 0.79 DRD2 (0.52) NPC1RAB9ASMN1; SMN2MAPTL3MBTL1
SCHEMBL13059256 0.79 NPC1 (0.58) NPC1RAB9ASMN1; SMN2HPGDMAPT
SCHEMBL7934205 0.78 KDM4E (0.49) NPC1RAB9ASMN1; SMN2HPGDMAPT
SCHEMBL14167586 0.77 CA2 (0.48) NPC1RAB9ASMN1; SMN2HPGDMAPT
SCHEMBL6339474 0.77 LTA4H (0.53) NPC1RAB9ASMN1; SMN2HPGDMAPT
SCHEMBL11285757 0.77 KCNA3 (0.58) NPC1RAB9AL3MBTL1ALDH1A1LMNA
SCHEMBL6397212 0.77 LTA4H (0.55) RAB9ATP53CYP1A2CYP3A4CYP2C9
SCHEMBL7934072 0.75 KDM4E (0.43) RAB9AMAPTL3MBTL1NQO1
SCHEMBL23267826 0.74 MEN1 (0.50) NPC1RAB9ASMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140896-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 Takeda Chemical Industries, Ltd. (JP) 2001-10-10 EP disclosed
US-6235771-B1 AIDS THERPAY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
WO-2000037455-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-06-29 WO disclosed