SCHEMBL7934216

SCHEMBL7934216

CCCOCCOc1ccc(OB(O)O)c(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.43
KDM4E B2RXH2 7/20 0.41
ALDH1A1 P00352 5/20 0.39
TDP1 Q9NUW8 4/20 0.39
CSNK2A1 P68400 2/20 0.38
MAPK1 P28482 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.35
LMNA P02545 2/20 0.35
RARB P10826 1/20 0.35
GLA P06280 1/20 0.35
ACACB O00763 1/20 0.35
MEN1 O00255 1/20 0.35
USP2 O75604 1/20 0.35
CYP3A4 P08684 1/20 0.35
CASP1 P29466 1/20 0.35
KMT2A Q03164 1/20 0.35
SLCO1B3 Q9NPD5 1/20 0.35
SLCO1B1 Q9Y6L6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7931128 0.89 L3MBTL1 (0.46) L3MBTL1KDM4EALDH1A1TDP1CSNK2A1
SCHEMBL7934212 0.89 L3MBTL1 (0.44) L3MBTL1KDM4EALDH1A1TDP1CSNK2A1
SCHEMBL7934233 0.84 KDM4E (0.40) L3MBTL1KDM4EALDH1A1TDP1MAPK1
SCHEMBL7928487 0.83 RARB (0.41) L3MBTL1KDM4EALDH1A1TDP1MAPK1
SCHEMBL7931127 0.80 L3MBTL1 (0.48) L3MBTL1KDM4EALDH1A1CSNK2A1SMN1; SMN2
SCHEMBL6344107 0.79 L3MBTL1 (0.47) L3MBTL1KDM4EALDH1A1TDP1CSNK2A1
SCHEMBL5657236 0.79 LMNA (0.45) L3MBTL1KDM4EALDH1A1MAPK1SMN1; SMN2
SCHEMBL7221364 0.77 ALDH1A1 (0.48) L3MBTL1KDM4EALDH1A1TDP1MAPK1
SCHEMBL7216146 0.76 HTR1A (0.40) L3MBTL1KDM4EALDH1A1TDP1SMN1; SMN2
SCHEMBL3787950 0.75 CSNK2A1 (0.62) L3MBTL1KDM4EALDH1A1TDP1CSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140896-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 Takeda Chemical Industries, Ltd. (JP) 2001-10-10 EP disclosed
US-6235771-B1 AIDS THERPAY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
WO-2000037455-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-06-29 WO disclosed