SCHEMBL7937232

SCHEMBL7937232

COC(=O)C(Sc1nc(C)cc(C)n1)C(C)(c1ccccc1)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.44
LMNA P02545 2/20 0.44
EDNRB P24530 4/20 0.43
EDNRA P25101 4/20 0.43
NR1I2 O75469 1/20 0.43
KCNE1 P15382 1/20 0.43
KCNQ1 P51787 1/20 0.43
POLB P06746 1/20 0.43
ALDH1A1 P00352 4/20 0.41
HPGD P15428 2/20 0.41
MAPT P10636 2/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 2/20 0.41
PKM P14618 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7934306 0.92 EDNRB (0.46) KDM4ELMNAEDNRBEDNRAALDH1A1
SCHEMBL7937196 0.86 EDNRB (0.49) EDNRBEDNRA
SCHEMBL8098308 0.75 EDNRB (0.50) EDNRBEDNRA
SCHEMBL7928120 0.75 EDNRB (0.44) KDM4ELMNAEDNRBEDNRAALDH1A1
SCHEMBL1069539 0.72 EDNRB (0.55) EDNRBEDNRANR1I2KCNE1KCNQ1
SCHEMBL7934325 0.72 MAPT (0.43) KDM4ELMNAEDNRBEDNRAPOLB
SCHEMBL7937185 0.72 EDNRA (0.44) KDM4ELMNAEDNRAPOLBALDH1A1
SCHEMBL8109239 0.72 EDNRB (0.57) EDNRBEDNRA
SCHEMBL8116655 0.69 EDNRB (0.46) EDNRBEDNRA
SCHEMBL1068997 0.69 KMT2A (0.50) ALDH1A1MAPTCYP1A2CYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235903-B1 Method for preparing sulfanyl-type endothelin receptor antagonists BASF AKTIENGESELLSCHAFT (DE) 2001-05-22 US disclosed