SCHEMBL7928120

SCHEMBL7928120

COC(=O)C(Sc1nc(OC)cc(OC)n1)C(C)(c1ccc(OC)cc1)c1ccc(OC)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 5/20 0.44
EDNRA P25101 5/20 0.44
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
NFKB1 P19838 1/20 0.40
RAB9A P51151 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
ALOX5 P09917 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
MAPT P10636 2/20 0.38
KIF11 P52732 1/20 0.38
RECQL P46063 2/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
ALOX15 P16050 1/20 0.37
APEX1 P27695 1/20 0.37
MAPK1 P28482 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7937196 0.89 EDNRB (0.49) EDNRBEDNRA
SCHEMBL7934373 0.85 ALOX5 (0.41) EDNRBEDNRASMN1; SMN2NPC1TP53
SCHEMBL7934306 0.82 EDNRB (0.46) EDNRBEDNRASMN1; SMN2MAPTALDH1A1
SCHEMBL8098308 0.79 EDNRB (0.50) EDNRBEDNRA
SCHEMBL8109239 0.77 EDNRB (0.57) EDNRBEDNRA
SCHEMBL1069539 0.76 EDNRB (0.55) EDNRBEDNRA
SCHEMBL7937232 0.75 KDM4E (0.44) EDNRBEDNRASMN1; SMN2MAPTALDH1A1
SCHEMBL7934325 0.73 MAPT (0.43) EDNRBEDNRASMN1; SMN2NPC1RAB9A
SCHEMBL8116655 0.72 EDNRB (0.46) EDNRBEDNRAALOX5
SCHEMBL8634830 0.71 EDNRB (0.35) EDNRBEDNRAALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235903-B1 Method for preparing sulfanyl-type endothelin receptor antagonists BASF AKTIENGESELLSCHAFT (DE) 2001-05-22 US disclosed