SCHEMBL7936378

SCHEMBL7936378

Nc1scc(-c2cccnc2)c1C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 2/20 0.52
ALDH1A1 P00352 2/20 0.51
HPGD P15428 2/20 0.51
MEN1 O00255 1/20 0.51
LMNA P02545 1/20 0.51
KMT2A Q03164 1/20 0.51
PRKCZ Q05513 1/20 0.51
MKNK1 Q9BUB5 4/20 0.48
MKNK2 Q9HBH9 4/20 0.48
ANO1 Q5XXA6 1/20 0.47
HSD17B10 Q99714 2/20 0.47
CYP2A6 P11509 2/20 0.46
KMO O15229 2/20 0.45
CYP19A1 P11511 3/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
TDO2 P48775 1/20 0.43
CYP2E1 P05181 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8196570 0.84 ALDH1A1 (0.62) ALDH1A1HPGDMEN1LMNAKMT2A
SCHEMBL1799330 0.84 KMT2A (0.69) ALDH1A1HPGDMEN1LMNAKMT2A
SCHEMBL8188234 0.81 KMT2A (0.65) ALDH1A1HPGDMEN1LMNAKMT2A
SCHEMBL689937 0.80 ALDH1A1 (0.77) ALDH1A1HPGDMEN1LMNAKMT2A
SCHEMBL27473744 0.78 ANO1 (0.56) GPR35ALDH1A1MEN1LMNAKMT2A
SCHEMBL27749754 0.76 HSD17B10 (0.63) GPR35ALDH1A1HPGDMEN1LMNA
SCHEMBL13838083 0.76 PRKCZ (0.61) ALDH1A1HPGDMEN1LMNAKMT2A
SCHEMBL28675027 0.75 KMO (0.51) GPR35ALDH1A1MEN1KMT2AMKNK1
SCHEMBL4932598 0.75 HSD17B10 (0.51) ALDH1A1HPGDMEN1LMNAKMT2A
SCHEMBL12465745 0.75 HSD17B10 (0.51) ALDH1A1HPGDMEN1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028193-A1 COMPOUNDS INCLUDING PIMELIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO disclosed
CN-101351453-A Heterocyclic amide compound and use thereof TAKEDA PHARMACEUTICAL (JP) 2009-01-21 CN disclosed
WO-2008063668-A1 HETEROBICYCLIC METALLOPROTEASE INHIBITORS ALANTOS PHARMACEUTICALS HOLDING, INC. (US) 2008-05-29 WO disclosed