SCHEMBL7937544

SCHEMBL7937544

COC(C=O)[C@H]1C(=O)N(CC(=O)O)CCN1C(=O)C(CC(=O)N1CCN(c2ccncc2)CC1)NC(=O)OC(C)OC(C)=O

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.34
ITGB3 P05106 12/20 0.33
ITGA2B P08514 12/20 0.33
ROCK2 O75116 1/20 0.32
DPP4 P27487 1/20 0.31
DPP8 Q6V1X1 1/20 0.31
DPP7 Q9UHL4 1/20 0.31
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
TSHR P16473 1/20 0.30
ITGAV P06756 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7403351 0.88 ITGB3 (0.40) CASP1ITGB3ITGA2BROCK2DPP4
SCHEMBL7403355 0.88 ITGB3 (0.40) CASP1ITGB3ITGA2BROCK2DPP4
SCHEMBL7937541 0.88 ITGB3 (0.40) CASP1ITGB3ITGA2BROCK2DPP4
SCHEMBL7372688 0.83 CASP1 (0.36) CASP1ITGB3ITGA2B
Hydrochloric Acid SCHEMBL7363298 0.78 ITGB3 (0.43) CASP1ITGB3ITGA2BCYP3A4CYP2D6
Hydrochloric Acid SCHEMBL7363292 0.78 ITGB3 (0.43) CASP1ITGB3ITGA2BCYP3A4CYP2D6
Hydrochloric Acid SCHEMBL7363302 0.78 ITGB3 (0.43) CASP1ITGB3ITGA2BCYP3A4CYP2D6
Hydrochloric Acid SCHEMBL7364908 0.78 ITGB3 (0.43) CASP1ITGB3ITGA2BCYP3A4CYP2D6
SCHEMBL7937529 0.78 RORC (0.35) CASP1ITGB3ITGA2B
SCHEMBL7937548 0.77 ITGB3 (0.34) CASP1ITGB3ITGA2BROCK2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242600-B1 ANTIISCHEMIC AGENTS, ANTICOAGULANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-06-05 US disclosed