SCHEMBL7937529

SCHEMBL7937529

COC(C=O)[C@H]1C(=O)N(CC(=O)O)CCN1C(=O)C(CC(=O)N1CCN(c2ccncc2)CC1)N(C)Cc1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RORC P51449 7/20 0.35
CASP1 P29466 1/20 0.34
ITGB3 P05106 2/20 0.34
ITGA2B P08514 2/20 0.34
ALDH1A1 P00352 2/20 0.33
MAPK1 P28482 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
TMEM97 Q5BJF2 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
LMNA P02545 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7367242 0.87 ITGB3 (0.42) RORCCASP1ITGB3ITGA2B
SCHEMBL7931599 0.87 ITGB3 (0.42) RORCCASP1ITGB3ITGA2B
SCHEMBL7931603 0.87 ITGB3 (0.42) RORCCASP1ITGB3ITGA2B
SCHEMBL7372688 0.86 CASP1 (0.36) CASP1ITGB3ITGA2B
SCHEMBL7937532 0.78 ITGB3 (0.34) RORCCASP1ITGB3ITGA2BMAPK1
SCHEMBL7937544 0.78 CASP1 (0.34) CASP1ITGB3ITGA2B
SCHEMBL7367244 0.77 RORC (0.36) RORCLMNA
Hydrochloric Acid SCHEMBL7364672 0.76 ITGB3 (0.44) ITGB3ITGA2B
SCHEMBL7372151 0.75 DPP4 (0.40) ITGB3ITGA2BALDH1A1HSD17B10
SCHEMBL7371269 0.74 ITGB3 (0.39) CASP1ITGB3ITGA2BTMEM97SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242600-B1 ANTIISCHEMIC AGENTS, ANTICOAGULANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-06-05 US disclosed