SCHEMBL7937867

SCHEMBL7937867

CCCNc1cc(N)c2nc(-c3nccs3)c(=O)n(C3CC3)c2n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.36
CYP1A2 P05177 6/20 0.36
CASP1 P29466 6/20 0.36
CASP7 P55210 6/20 0.36
HSD17B10 Q99714 6/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
CYP2D6 P10635 2/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 6/20 0.35
HIF1A Q16665 3/20 0.35
CLK4 Q9HAZ1 2/20 0.34
MAPK1 P28482 2/20 0.34
USP2 O75604 2/20 0.34
AKT1 P31749 5/20 0.33
MTOR P42345 5/20 0.33
CYP2C9 P11712 2/20 0.33
BRD4 O60885 1/20 0.33
BRD2 P25440 1/20 0.33
BRD3 Q15059 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7945987 0.95 TYRO3 (0.36) ALDH1A1CYP1A2CASP1CASP7HSD17B10
SCHEMBL7947006 0.88 ALDH1A1 (0.34) ALDH1A1CYP1A2CASP1CASP7HSD17B10
SCHEMBL7944716 0.87 CYP1A2 (0.39) ALDH1A1CYP1A2CASP1CASP7HSD17B10
SCHEMBL7944000 0.85 ALDH1A1 (0.33) ALDH1A1CYP1A2CASP1CASP7HSD17B10
SCHEMBL7944790 0.85 ADORA2A (0.37) ALDH1A1CYP1A2HSD17B10CYP2D6LMNA
SCHEMBL7937747 0.84 HSF1 (0.35) ALDH1A1CYP1A2CASP1CASP7HSD17B10
SCHEMBL7938052 0.83 CCND1 (0.38) ALDH1A1CYP1A2CASP1CASP7HSD17B10
SCHEMBL7938054 0.82 AKT1 (0.41) ALDH1A1CYP1A2CASP1CASP7HSD17B10
SCHEMBL7938346 0.82 ALDH1A1 (0.38) ALDH1A1CYP1A2CASP1CASP7HSD17B10
SCHEMBL7945868 0.79 CYP1A2 (0.41) ALDH1A1CYP1A2CASP1CASP7HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008775-A1 AMINOPYRIDOPYRAZINONE DERIVATIVES FOR TREATING NEURODEGENERATIVE DISEASES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed