SCHEMBL7937747

SCHEMBL7937747

CCCNc1cc(N)c2nc(-c3nccs3)c(=O)n(CCC)c2n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSF1 Q00613 1/20 0.35
ADORA1 P30542 2/20 0.33
PDE7A Q13946 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33
LYN P07948 1/20 0.33
HPGD P15428 4/20 0.31
TLR7 Q9NYK1 1/20 0.31
MEN1 O00255 2/20 0.30
USP2 O75604 2/20 0.30
CYP1A2 P05177 2/20 0.30
CYP3A4 P08684 2/20 0.30
CYP2D6 P10635 2/20 0.30
MAPK1 P28482 2/20 0.30
CASP1 P29466 2/20 0.30
CASP7 P55210 2/20 0.30
KMT2A Q03164 2/20 0.30
HSD17B10 Q99714 2/20 0.30
CLK4 Q9HAZ1 2/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7943995 0.93 HSF1 (0.36) HSF1ADORA1PDE7AADORA3ADORA2A
SCHEMBL7944574 0.90 HSF1 (0.36) HSF1ADORA1ADORA3ADORA2ALYN
SCHEMBL7937752 0.85 ADORA2A (0.39) HSF1ADORA1ADORA3ADORA2ALYN
SCHEMBL7944078 0.80 PDE4B (0.42) HSF1ADORA1ADORA3ADORA2AMEN1
SCHEMBL7945987 0.79 TYRO3 (0.36) HSF1HPGDMEN1USP2CYP1A2
SCHEMBL7937864 0.77 ADORA2A (0.38) ADORA1PDE7AADORA3ADORA2ALYN
SCHEMBL7946794 0.75 ADORA1 (0.39) HSF1ADORA1PDE7AADORA3ADORA2A
SCHEMBL7945503 0.75 TLR9 (0.37) ADORA1ADORA2AHPGDCYP1A2CYP2D6
SCHEMBL7944114 0.74 PDE4B (0.48) HSF1ADORA1ADORA3ADORA2AHPGD
SCHEMBL7946084 0.72 HRH4 (0.37) ADORA1ADORA2AHPGDCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008775-A1 AMINOPYRIDOPYRAZINONE DERIVATIVES FOR TREATING NEURODEGENERATIVE DISEASES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed