SCHEMBL7939173

SCHEMBL7939173

N#Cc1ccc(COC(=O)Cc2cnc[nH]2)cc1

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.58
CYP19A1 P11511 5/20 0.46
ALDH1A1 P00352 2/20 0.44
CYP3A4 P08684 1/20 0.44
GABRA1 P14867 1/20 0.44
TSHR P16473 1/20 0.44
NFKB1 P19838 1/20 0.44
GABRR1 P24046 1/20 0.44
GABRR2 P28476 1/20 0.44
GABRA5 P31644 1/20 0.44
GABRB2 P47870 1/20 0.44
GABRA4 P48169 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
KDM4E B2RXH2 1/20 0.43
MAPT P10636 1/20 0.43
PMP22 Q01453 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL7939566 0.99 HRH3 (0.57) HRH3CYP19A1ALDH1A1CYP3A4GABRA1
SCHEMBL7704752 0.80 DAO (0.40) HRH3ALDH1A1CYP3A4GABRA1TSHR
SCHEMBL7924408 0.74 HRH3 (1.00) HRH3CYP19A1CYP3A4MAPT
SCHEMBL7468703 0.73 HRH3 (0.73) HRH3CYP19A1
SCHEMBL7505800 0.71 HRH3 (0.54) HRH3CYP19A1
SCHEMBL6669234 0.71 GAA (0.48) ALDH1A1TSHRTDP1
SCHEMBL31377271 0.71 ALDH1A1 (0.58) HRH3ALDH1A1CYP3A4GABRA1TSHR
SCHEMBL10569744 0.70 ALDH1A1 (0.51) ALDH1A1CYP3A4KDM4EMAPT
SCHEMBL3716431 0.70 HTT (0.53) ALDH1A1TSHRTDP1
SCHEMBL7703566 0.70 HRH3 (0.68) HRH3CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001017992-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-03-15 WO disclosed