SCHEMBL793965

SCHEMBL793965

CC(C)COC(=O)N1CCC(Nc2cc(C=O)cc(Nc3nc4cccnc4s3)n2)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 5/20 0.56
LCK P06239 3/20 0.47
AURKB Q96GD4 3/20 0.47
NOS2 P35228 5/20 0.44
NOS1 P29475 4/20 0.41
NOS3 P29474 2/20 0.41
RORC P51449 1/20 0.40
DHODH Q02127 1/20 0.40
SSTR5 P35346 1/20 0.40
HCK P08631 2/20 0.38
BTK Q06187 2/20 0.38
PDE10A Q9Y233 2/20 0.37
MAP4K4 O95819 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
ATM Q13315 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL793964 0.87 ITK (0.56) ITKLCKAURKBNOS2RORC
SCHEMBL807716 0.82 ITK (0.60) ITKLCKAURKBRORCDHODH
SCHEMBL2371312 0.81 ITK (0.62) ITKLCKAURKBBTKSMN1; SMN2
SCHEMBL2371318 0.81 ITK (0.62) ITKLCKAURKBBTKSMN1; SMN2
SCHEMBL3578949 0.76 NOS2 (0.61) NOS2NOS1NOS3RORCDHODH
Hydrochloric Acid SCHEMBL9774607 0.76 NOS2 (0.60) NOS2NOS1NOS3RORCDHODH
SCHEMBL807541 0.74 ITK (0.55) ITKLCKAURKBRORCDHODH
SCHEMBL2394365 0.73 ITK (0.61) ITKLCKAURKBSSTR5BTK
SCHEMBL2394354 0.73 ITK (0.61) ITKLCKAURKBSSTR5BTK
SCHEMBL807822 0.72 ITK (0.81) ITKLCKAURKBRORCDHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035055-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-22 WO disclosed