SCHEMBL807716

SCHEMBL807716

CC(C)(C)OC(=O)N1CC[C@H](Nc2cc(C=O)cc(Nc3nc4cccnc4s3)n2)C1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITK Q08881 2/20 0.60
BTK Q06187 6/20 0.42
HCK P08631 5/20 0.42
ADORA3 P0DMS8 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA2B P29275 1/20 0.41
LCK P06239 1/20 0.41
AURKB Q96GD4 1/20 0.41
USP30 Q70CQ3 4/20 0.41
CCNA2 P20248 1/20 0.40
CDK2 P24941 1/20 0.40
PIM1 P11309 2/20 0.39
PIM2 Q9P1W9 2/20 0.39
SYK P43405 1/20 0.39
RORC P51449 1/20 0.39
DHODH Q02127 1/20 0.39
PIK3CD O00329 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL793964 0.95 ITK (0.56) ITKBTKHCKLCKAURKB
SCHEMBL807822 0.85 ITK (0.81) ITKBTKHCKADORA3ADORA2A
SCHEMBL807926 0.85 ITK (0.59) ITKBTKHCKADORA3ADORA2A
SCHEMBL807803 0.84 ITK (0.58) ITKBTKHCKADORA3ADORA2A
SCHEMBL793965 0.82 ITK (0.56) ITKBTKHCKLCKAURKB
SCHEMBL807541 0.80 ITK (0.55) ITKLCKAURKBCCNA2CDK2
SCHEMBL2371318 0.78 ITK (0.62) ITKBTKLCKAURKB
SCHEMBL2371312 0.78 ITK (0.62) ITKBTKLCKAURKB
SCHEMBL20767484 0.75 ITK (1.00) ITKBTKHCKLCKAURKB
SCHEMBL20767486 0.75 ITK (1.00) ITKBTKHCKLCKAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035055-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-22 WO disclosed