SCHEMBL807822

SCHEMBL807822

C[C@H](NCc1cc(Nc2nc3cccnc3s2)nc(NC2CCN(C(=O)OC(C)(C)C)C2)c1)C(C)(C)C

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 2/20 0.81
ADORA2A P29274 2/20 0.41
ADORA2B P29275 2/20 0.41
ADORA3 P0DMS8 1/20 0.41
LCK P06239 1/20 0.41
AURKB Q96GD4 1/20 0.41
HCK P08631 2/20 0.38
BTK Q06187 2/20 0.38
USP30 Q70CQ3 5/20 0.38
RORC P51449 1/20 0.38
DHODH Q02127 1/20 0.38
SSTR5 P35346 1/20 0.37
CCNA2 P20248 1/20 0.37
CDK2 P24941 1/20 0.37
PIM1 P11309 2/20 0.36
PIM2 Q9P1W9 2/20 0.36
SYK P43405 1/20 0.36
BRD4 O60885 1/20 0.36
CCNT1 O60563 1/20 0.36
PIK3CD O00329 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20767484 0.90 ITK (1.00) ITKLCKAURKBHCKBTK
SCHEMBL20767486 0.90 ITK (1.00) ITKLCKAURKBHCKBTK
SCHEMBL20767487 0.90 ITK (1.00) ITKLCKAURKBHCKBTK
SCHEMBL25069003 0.86 ITK (0.76) ITKLCKAURKBHCKBTK
SCHEMBL23409058 0.86 ITK (0.76) ITKLCKAURKBHCKBTK
SCHEMBL25069001 0.85 ITK (0.75) ITKLCKAURKBHCKBTK
SCHEMBL25069002 0.85 ITK (0.75) ITKLCKAURKBHCKBTK
SCHEMBL807716 0.85 ITK (0.60) ITKADORA2AADORA2BADORA3LCK
SCHEMBL807926 0.85 ITK (0.59) ITKADORA2AADORA2BADORA3LCK
SCHEMBL807803 0.84 ITK (0.58) ITKADORA2AADORA2BADORA3LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035055-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-22 WO disclosed