SCHEMBL7940291

SCHEMBL7940291

C#Cc1c(C)cc(C)cc1Cc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39
BCL2 P10415 1/20 0.39
BCL2L1 Q07817 1/20 0.39
IDH1 O75874 2/20 0.36
PDE2A O00408 1/20 0.36
GPR55 Q9Y2T6 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
CALM1 P0DP23 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2A6 P11509 1/20 0.35
ALOX5 P09917 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
LDHA P00338 1/20 0.35
LDHB P07195 1/20 0.35
C5AR1 P21730 1/20 0.34
MEN1 O00255 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzene SCHEMBL7940296 0.75 RAPGEF4 (0.36) TSHRCYP1A2CYP2A6
SCHEMBL544660 0.74 BCL2 (0.52) BCL2BCL2L1ALOX5LDHALDHB
SCHEMBL30292338 0.71 TP53 (0.35) CYP3A4CYP2D6TSHRCYP2C19BCL2
SCHEMBL1062516 0.71 RAPGEF4 (0.39) TSHRCYP1A2CYP2A6HSD17B10
SCHEMBL1276089 0.71 CYP3A4 (0.57) CYP3A4CYP2D6TSHRCYP2C19BCL2
SCHEMBL670158 0.71 BCL2 (0.57) CYP2C19BCL2BCL2L1ALOX5HIF1A
SCHEMBL3301748 0.71 CYP3A4 (0.53) CYP3A4CYP2D6TSHRCYP2C19BCL2
SCHEMBL28049389 0.71 BCL2 (0.47) CYP3A4CYP2D6TSHRCYP2C19BCL2
SCHEMBL7819859 0.70 CALM1 (0.48) CYP3A4CYP2D6TSHRCYP2C19BCL2
SCHEMBL12816424 0.70 CYP3A4 (0.39) CYP3A4CYP2D6TSHRCYP2C19BCL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288279-B1 THEIR PREPARATION PROCESS AND THEIR USE IN ASYMMETRICAL CATALYSIS. REARRANGING A DIPHOSPHOLE, REACTING THE DIPHOSPHOLE WITH AN ACETYLENIC COMPOUND TO FORM THE DIPHOSPHINE RHODIA CHIMIE (FR) 2001-09-11 US claimed