SCHEMBL7941853

SCHEMBL7941853

CC(=O)Oc1ccc2c(=O)c(-c3ccccc3)c(C)oc2c1OC(C)=O

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.69
ALDH1A1 P00352 7/20 0.69
MAPT P10636 6/20 0.69
GAA P10253 5/20 0.69
SMN1; SMN2 Q16637 3/20 0.69
HPGD P15428 3/20 0.69
LMNA P02545 2/20 0.69
MPI P34949 1/20 0.69
POLB P06746 2/20 0.56
RECQL P46063 2/20 0.56
PKM P14618 1/20 0.56
HTT P42858 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
ADORA3 P0DMS8 5/20 0.54
ADORA2A P29274 2/20 0.54
ADORA1 P30542 2/20 0.54
CYP3A4 P08684 1/20 0.46
HSD17B10 Q99714 2/20 0.46
GLA P06280 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12941614 0.88 GAA (0.58) KDM4EALDH1A1MAPTGAASMN1; SMN2
SCHEMBL27459594 0.88 KDM4E (0.55) KDM4EALDH1A1MAPTGAASMN1; SMN2
SCHEMBL7912397 0.85 ADORA3 (0.59) KDM4EALDH1A1MAPTGAASMN1; SMN2
SCHEMBL8123765 0.84 ADORA3 (0.60) KDM4EALDH1A1MAPTGAASMN1; SMN2
SCHEMBL10939957 0.81 KDM4E (0.67) KDM4EALDH1A1MAPTGAASMN1; SMN2
SCHEMBL1628395 0.80 ALDH1A1 (0.67) KDM4EALDH1A1MAPTGAASMN1; SMN2
SCHEMBL6617327 0.79 MAPT (0.60) KDM4EALDH1A1MAPTGAASMN1; SMN2
SCHEMBL30233473 0.79 MAPT (0.60) KDM4EALDH1A1MAPTGAASMN1; SMN2
SCHEMBL10995103 0.78 KDM4E (0.62) KDM4EALDH1A1MAPTGAASMN1; SMN2
SCHEMBL31619650 0.76 KDM4E (0.59) KDM4EALDH1A1MAPTGAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6255497-B1 DAIDZIN DERIVATIVES AS ENZYME INHIBITORS OF ALDEHYDE DEHYDROGENASE; USEFUL IN TREATING ALCOHOLISM THE ENDOWMENT FOR RESEARCH IN HUMAN BIOLOGY, INC. 2001-07-03 US disclosed
EP-0592583-A1 METHOD FOR THE INHIBITION OF ALDH-I USEFUL IN THE TREATMENT OF ALCOHOL DEPENDENCE OR ALCOHOL ABUSE THE ENDOWMENT FOR RESEARCH IN HUMAN BIOLOGY, INC. (US) 1994-04-20 EP disclosed
WO-1993000896-A1 METHOD FOR THE INHIBITION OF ALDH-I USEFUL IN THE TREATMENT OF ALCOHOL DEPENDENCE OR ALCOHOL ABUSE THE ENDOWMENT FOR RESEARCH IN HUMAN BIOLOGY, INC. (US) 1993-01-21 WO disclosed