SCHEMBL7943341

SCHEMBL7943341

COc1cc(-c2ccc(C(F)(F)F)cc2)ccc1CO

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 2/20 0.52
CD274 Q9NZQ7 2/20 0.52
KIF11 P52732 2/20 0.50
AKR1C3 P42330 1/20 0.45
AKR1C2 P52895 1/20 0.45
MGAM O43451 3/20 0.43
GAA P10253 3/20 0.43
SI P14410 3/20 0.43
MGAM2 Q2M2H8 3/20 0.43
MCHR1 Q99705 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.41
IDO1 P14902 1/20 0.41
TDO2 P48775 1/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 1/20 0.41
CTSA P10619 1/20 0.41
CASR P41180 2/20 0.40
BACE1 P56817 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6498758 0.87 PDCD1 (0.46) PDCD1CD274GAAMEN1KMT2A
SCHEMBL31321848 0.87 PDCD1 (0.46) PDCD1CD274GAAMEN1KMT2A
SCHEMBL12650491 0.86 KIF11 (0.55) KIF11AKR1C3AKR1C2MGAMGAA
SCHEMBL8021476 0.83 S1PR1 (0.52) PDCD1CD274KIF11
SCHEMBL7935451 0.82 PPARD (0.43) KIF11MCHR1KMT2ABACE1
SCHEMBL8028294 0.80 PDCD1 (0.58) PDCD1CD274MEN1KMT2AALDH1A1
SCHEMBL6497164 0.80 PDCD1 (0.62) PDCD1CD274GAAKMT2AALDH1A1
SCHEMBL25688156 0.80 CYP1A2 (0.49) GAAMEN1KMT2AALDH1A1
SCHEMBL25688144 0.80 AKR1C3 (0.47) PDCD1CD274AKR1C3AKR1C2MEN1
SCHEMBL1779625 0.79 RXRA (0.54) KIF11MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010015653-A1 PYRIMIDINE DERIVATIVES AS ACTIVATORS OF SOLUBLE GUANYLATE CYCLASE SMITHKLINE BEECHAM CORPORATION (US) 2010-02-11 WO disclosed
WO-2009071504-A1 2,6-DISUBSTITUTED PYRIDINES AS SOLUBLE GUANYLATE CYCLASE ACTIVATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-06-11 WO disclosed